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2-{4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-1-yl}phenol
5-[({[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
2-methyl-6-{2-[4-phenyl-5-(1,3-thiazol-2-yl)-1H-imidazol-1-yl]ethyl}pyrimidin-4-ol
2-{3-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]phenoxy}propanamide
2-[(1S,5R)-3-[(2-chloro-4-fluorophenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
8-(3-chloro-4-hydroxybenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3,6-diazabicyclo[3.2.2]nonane
3-ethyl-4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1H-pyrazole
4-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]-N-methylbenzamide
3-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)carbamoyl}amino)-4-methyl-N-propylbenzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-{[7-fluoro-2-(thiophen-2-yl)quinolin-3-yl]methyl}acetamide
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(pyrazin-2-yl)propanamide
N-[(1-{[1-(propan-2-yl)-1H-pyrrol-3-yl]methyl}pyrrolidin-3-yl)methyl]pyridine-4-carboxamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(2-methyl-1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-methyl-2-{2-[(2-methyl-6-propylpyrimidin-4-yl)amino]ethyl}-3,4-dihydropyrimidin-4-one
N'-(3,5-dimethylphenyl)-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]propanediamide
1-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(3,4,5-trimethoxyphenyl)-1H-imidazole
2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-3-phenylcycloprop-2-ene-1-carboxamide
N-[(2-fluorophenyl)methyl]-4-(4-{[2-methyl-2-(morpholin-4-yl)propyl]amino}piperidin-1-yl)benzamide
1-(diphenylmethyl)-N-[(5-methylpyrazin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-(4-hydroxyphenyl)-2-phenyl-N-[2-(piperidin-1-yl)ethyl]propanamide
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-(2-hydroxy-2-phenylethyl)-1,3-oxazole-4-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(thiophen-2-yl)acetyl]pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
1-(azocan-1-yl)-3-[2-methoxy-4-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
1-(2-benzylmorpholin-4-yl)-2-(methylsulfanyl)ethan-1-one
2-ethoxy-5-(2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}pyrimidin-4-yl)benzoic acid
2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-(2-oxopyrrolidin-1-yl)propanamide
(2S)-N-{1-[(3-methylphenyl)methyl]cyclopropyl}-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
methyl 4-[({[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]benzoate
5-[(3,5-difluorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-(1-hydroxybutan-2-yl)-N-(thiophen-2-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide
3-({[7-fluoro-1-(2-methylpropyl)-2-oxo-1,2-dihydroquinolin-3-yl]methyl}amino)-1λ6-thiolane-1,1-dione
2-[2-(dimethylamino)ethyl]-8-[(3E)-pent-3-enoyl]-2,8-diazaspiro[5.5]undecan-3-one
[4-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1,4-oxazepan-6-yl]methanol
2-methoxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}benzene-1-sulfonamide
3-(3-methoxyphenyl)-N-{[5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
3-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1H-indole
2-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-2,3-dihydro-1H-isoindole
8-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2,3,5,6-tetramethylbenzamide
(3R,5S)-5-(1-cyclohexyl-3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-3-ol
3-acetamido-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
(3S,4R)-1-[2-(methylsulfanyl)acetyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-ethyl-3,5-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-indole-2-carboxamide
(1S,5R)-3-[2-(2,3-dimethoxyphenyl)acetyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-N-[4-(furan-2-yl)phenyl]piperidine-3-carboxamide
1-methoxy-3-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)propan-2-ol