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7-[2-(1H-1,3-benzodiazol-1-yl)propanoyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 5-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]-1H-imidazole-4-carboxylate
3-cyclohexyl-1-[4-(difluoromethoxy)phenyl]-3-(pyridin-2-ylmethyl)urea
3,4,7-trimethyl-2-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1H-indole
2-(dimethylamino)-N-[1-(3-methylbutanoyl)piperidin-4-yl]-2-(2-methylphenyl)acetamide
3-methyl-9-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}-3,9-diazaspiro[5.6]dodecane
(2-ethoxy-5-{[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methyl}phenyl)methanol
(3R,5R)-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-methyl-6-oxopiperidine-3-carboxamide
4-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
1-(3,5-dimethyl-1H-indole-2-carbonyl)-N-[2-(dimethylamino)ethyl]-N-methylpiperidin-3-amine
N-(4-chloronaphthalen-1-yl)-3-(piperidin-1-yl)pyrrolidine-1-carboxamide
2-(6-chloropyridin-3-yl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
(2R,6R)-4-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-(1-ethylpiperidin-4-yl)-N-methyl-N-[1-(pyridin-3-yl)propyl]acetamide
2-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-6-methyl-4H-pyran-4-one
2-(1H-imidazole-5-carbonyl)-6-methyl-5-[5-(1-methylpyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-({1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
methyl 3-(cyclobutylmethoxy)-5-[methyl(pyridin-2-ylmethyl)carbamoyl]benzoate
2-(methylamino)-N-{2-[(pyridin-3-yl)amino]ethyl}pyridine-4-carboxamide
{1-[1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)piperidin-4-yl]ethyl}dimethylamine
2-(cyclopentylmethyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
6-methoxy-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-4-amine
(2S,4S)-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
5-ethyl-N-[(4-sulfamoylphenyl)methyl]thiophene-2-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3-(2-methylphenyl)-3-phenylpropanamide
[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carbonitrile
2-(4-{1-[1-(propan-2-yl)piperidin-4-yl]pyrrolidin-3-yl}piperidin-1-yl)pyrimidine
3-[(3R,4S)-4-(dimethylamino)-1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-3-yl]propanoic acid
4-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)piperazine-1-carboxamide
5-[(2S)-1-acetylpyrrolidine-2-carbonyl]-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-N-[2-(morpholin-4-yl)ethyl]pyridin-2-amine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-ethylpiperidine-4-carboxamide
N-(1-methanesulfonylpiperidin-4-yl)-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
5-[5-(3,5-dimethyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
2-{4-[6-amino-5-cyano-4-(pyridin-3-yl)pyridin-2-yl]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
(2E)-N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-2-yl)prop-2-enamide
2-({4-[(3,5-dimethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methyl-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
9-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]propanoic acid
2-(phenylsulfanyl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-methyl-3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-1,2,5,6,7,8-hexahydroquinolin-2-one
N-[2-(propylsulfanyl)ethyl]piperidin-3-amine
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
2-(dimethylamino)-7-(oxolane-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-ethyl-8-[(4-methoxyphenyl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione