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N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-4-(1H-pyrazol-1-yl)benzamide
1-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-{3-[4-(2-methylpropoxy)phenyl]-1H-pyrazole-5-carbonyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-2,3-dihydro-1H-inden-2-amine
1-methyl-4-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}pyrrolidin-2-one
2-(2,3-dihydro-1H-inden-1-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
N-{4-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]phenyl}cyclobutanecarboxamide
3-cyclohexyl-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
4-(2,3-dihydro-1H-inden-2-yl)-11-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
8-(2-amino-6-methylpyrimidin-4-yl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 3-methoxy-5-[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})carbamoyl]benzoate
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-methylpyrimidine-5-carbonyl)piperidin-3-ol
5-(3-methyl-1,2,4-oxadiazol-5-yl)-2-[4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine
1-{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-3-ol
4-{[2-(dimethylamino)ethyl]amino}-5-methyl-N-{[4-(trifluoromethyl)phenyl]methyl}thieno[2,3-d]pyrimidine-6-carboxamide
1-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
3-(prop-2-en-1-yloxy)-N-[(1r,4r)-4-hydroxycyclohexyl]benzamide
N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-1H-imidazole-2-carboxamide
(1R,3S)-3-ethoxy-7-(5-hydroxypyrazine-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
3-(2,5-dioxoimidazolidin-4-yl)-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}propanamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-(2-oxopiperidin-1-yl)acetamide
N-[2-(4-{[(4-methylphenyl)methyl]carbamoyl}-1H-1,2,3-triazol-1-yl)ethyl]pyridine-2-carboxamide
1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-[2-(4-fluorophenyl)-1-{1-[2-(3-methoxyphenyl)acetyl]piperidin-4-yl}ethyl]-2-methoxy-N-methylacetamide
2-{9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carbonyl}benzonitrile
3-({1-[(dimethylcarbamoyl)methyl]piperidin-4-yl}methyl)benzoic acid
(3S,4S)-3-hydroxy-4-(morpholin-4-yl)-N-[4-(1H-pyrazol-1-yl)phenyl]pyrrolidine-1-carboxamide
5-amino-1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pentan-1-one
4-[5-(hydroxymethyl)furan-2-carbonyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
8-(1H-indol-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(1-methyl-1H-pyrazol-4-yl)methyl][(3-methyl-1H-pyrazol-5-yl)methyl](2-methylpropyl)amine
1-(3-cyanophenyl)-3-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-5-methylpyrazine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(furan-3-carbonyl)piperidine-3-carboxylate
9-methoxy-4-[(3-methoxyphenyl)methyl]-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){[2-(morpholin-4-yl)quinolin-3-yl]methyl}amine
4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-6-ethyl-2-methylquinoline
3-(propan-2-yl)-5-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]pyrrolidin-2-yl}-1,2,4-oxadiazole
(3S,5R)-1-(pyridin-4-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
2-(trifluoromethyl)-4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]morpholine
1-tert-butyl-3-cyclopropyl-5-[2-(ethylsulfanyl)ethyl]-1H-1,2,4-triazole
N-{[1-(1H-indol-2-ylmethyl)piperidin-4-yl]methyl}pyridazine-3-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}cyclopropanecarboxamide
3-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-1H-indazole
3-(2-ethyl-1H-imidazol-1-yl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
N-cyclopropyl-1-[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-[3-(morpholine-4-carbonyl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one