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5-methyl-1-{2-oxo-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-4-[3-(2-methylphenoxymethyl)piperidine-1-carbonyl]pyridin-2-amine
(4aS,8aR)-1-(3-aminopropyl)-6-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
3-(1-methyl-1H-pyrrol-2-yl)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
N-cyclopropyl-4-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperazine-2-carboxamide
N-methyl-N-(3-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-3-oxopropyl)methanesulfonamide
N-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-N-methyloxolan-3-amine
N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-5-propyl-1,2-oxazole-4-carboxamide
N-benzyl-1-[1-(but-3-enoyl)piperidin-4-yl]piperidine-3-carboxamide
1-(3-{4-[(4-fluorophenyl)amino]piperidin-1-yl}phenyl)-3-methylimidazolidin-2-one
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-imidazol-1-yl)propyl]acetamide
1-(5-chloropyridin-2-yl)-4-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazine
4-chloro-1-methyl-5-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1H-pyrazole
3-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
(1S,5R)-3-methyl-6-(3-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
2,2-dimethyl-1-(thiophen-2-yl)-N-(4H-1,2,4-triazol-4-yl)cyclopropane-1-carboxamide
N,N-diethyl-7,8-dimethyl-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
[(3,5-difluoro-4-methoxyphenyl)methyl](methyl)[1-(pyridin-4-yl)ethyl]amine
1-{[4-(3-ethoxyphenoxy)-3-methoxyphenyl]methyl}pyrrolidine
N-cyclopropyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
2-{[4-(4-chloro-2-methylphenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]propanamide
N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
2-methoxy-2-methyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}propanamide
(4aR,7aS)-1-acetyl-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-fluoro-5-methylphenyl)-N'-[2-methoxy-1-(pyridin-2-yl)ethyl]butanediamide
1-ethyl-4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]piperazine
2-(azepane-1-carbonyl)-6-(4-methoxyphenyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]oxane-2-carboxamide
(1R,2R)-N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-2-phenylcyclopropane-1-carboxamide
3-cyano-N-(3,5-difluorophenyl)piperidine-1-carboxamide
N-(2-acetamidophenyl)-2-{[1-(3-methylpyridin-2-yl)propan-2-yl]amino}acetamide
(1-benzothiophen-2-ylmethyl)({[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
3-[1-(6-chloropyridazin-3-yl)piperidin-3-yl]-1-[2-(dimethylamino)ethyl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(5-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
4-{[5-(4-ethyl-1,2,3-thiadiazol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-propylpiperidine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
4-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
3-(methoxymethyl)-1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidine
N-(3-methylbutyl)-5-[1-(1,2,3-thiadiazole-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
5-methyl-2-[3-(thiomorpholin-4-ylmethyl)phenyl]-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
5-(2,6-difluorophenoxymethyl)-N-[1-(1H-indol-1-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
3,6-dimethyl-4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-[1,2]oxazolo[5,4-b]pyridine
[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})(propan-2-yl)amine
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-[(6-methylpyridin-2-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[4-(7-chloro-1-methyl-1H-indole-2-carbonyl)morpholin-3-yl]acetic acid
N-benzyl-4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]amine
N-cyclohexyl-5-cyclopropyl-N-(2-hydroxy-2-phenylethyl)-1H-pyrazole-3-carboxamide