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1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
4-[(3-{2-tert-butylimidazo[1,2-a]pyrimidin-3-yl}phenyl)methyl]morpholine
1-(thiophen-2-ylmethyl)-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
6-{[(4-fluorophenyl)methyl](methyl)amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
(3R,9aR)-8-(2,3-difluorobenzoyl)-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{2-[2-(trifluoromethyl)phenyl]ethyl}pyrimidin-4-amine
3-(3-methoxyphenyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2,2-dimethylpropanamide
N-[(4-hydroxyazepan-4-yl)methyl]-4-methyl-2-phenylpyrimidine-5-carboxamide
2-[2-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1H-imidazol-1-yl]acetamide
4-({2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)-1-phenyl-1H-1,2,3-triazole
[2-(azepan-1-yl)ethyl][(2,5-difluorophenyl)methyl]ethylamine
N-phenyl-5-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]pyrimidin-2-amine
1-[(4-fluorophenyl)methyl]-4-(6-methylpyridazin-3-yl)-1,4-diazepane
4-[4-methyl-5-(5-methylthiophen-2-yl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
8-methoxy-N-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-amine
4-[(2-chlorophenyl)methyl]-1-[(2,4-difluorophenyl)methyl]-1,4-diazepan-5-one
1-[(2-ethylpyrimidin-5-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
(3R,4R)-1-(5-chloropyridin-2-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
2-ethoxy-1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]ethan-1-one
5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrazin-2-ol
(3aR,6aR)-2-benzyl-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
{2-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}urea
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(1H-indol-4-ylmethyl)benzamide
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-2-carbonitrile
(2S,4S)-4-amino-1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-{[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]sulfamoyl}-N-phenylbenzamide
4-[(3-fluorophenyl)methyl]-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1S,2R)-N1-[3-(morpholin-4-yl)propyl]-N2-propylcyclohexane-1,2-dicarboxamide
1,3-dimethyl-4-[5-(trifluoromethyl)pyridin-2-yl]piperazin-2-one
3-(2-methylpropyl)-N-[2-(1H-pyrrol-1-yl)ethyl]-1,2-oxazole-5-carboxamide
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-dimethyl-1-benzofuran-2-carboxamide
(2S,4R)-N-[2-(2-fluorophenyl)ethyl]-4-[(naphthalen-1-ylmethyl)amino]-1-(propan-2-yl)pyrrolidine-2-carboxamide
3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(piperidin-1-yl)ethan-1-one
2-{1-[(4-fluorophenyl)methyl]-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-3-methylbenzene-1-sulfonamide
2-hydroxy-3-(2-methylphenoxy)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
N-[3-(hydroxymethyl)-2-methylphenyl]-4-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}benzamide
[(3-chloropyridin-4-yl)methyl](methyl)[(3-methylpyridin-2-yl)methyl]amine
(3aS,7aR)-2-[5-(ethylsulfanyl)thiophene-2-carbonyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
9-(5-methoxyfuran-2-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-(thiophen-3-ylmethyl)benzamide
5-(4-fluorophenyl)-N-[3-(1H-imidazol-1-yl)propyl]-1,2,4-triazin-3-amine
1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)cyclopropan-1-amine
2-ethoxy-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyridine
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2-(4-propanoylphenoxy)acetamide