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4-[1-(4-methyl-2-phenylpyrimidine-5-carbonyl)piperidin-4-yl]thiomorpholine
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)ethan-1-one
5-(3-benzylpyrrolidine-1-carbonyl)-1-methyl-3-(2-methylpropyl)-1H-pyrazole
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
(3S,4S)-1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-4-(dimethylamino)pyrrolidin-3-ol
methyl (2S)-1-(4-{[2-(1H-indol-3-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidine-2-carboxylate
5-amino-1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pentan-1-one
3-chloro-N-(cyclopropylmethyl)-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
4-{[({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)amino]methyl}-1,2-dihydrophthalazin-1-one
3-chloro-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}pyridin-2-amine
N-(1-{[methyl(2-methylpropyl)carbamoyl]methyl}-1H-pyrazol-4-yl)pyridine-2-carboxamide
2-methyl-5-{4-[3-(1H-pyrazol-1-yl)phenyl]phenyl}-1,3,4-oxadiazole
1-(4-{2-[3-(3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
N-butyl-3-[3-(trifluoromethyl)benzoyl]piperidine-1-carboxamide
(3S,4S)-1-[2-chloro-5-(trifluoromethyl)benzoyl]-4-methylpiperidine-3,4-diol
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]urea
N-[(3R,4R)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-(pyridin-3-yl)morpholine
4-fluoro-3-[2-(furan-2-yl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
5-methyl-14-[(1E)-1-phenylprop-1-en-2-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(2S)-2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-4-(methylsulfanyl)butan-1-ol
N-benzyl-N-[2-(dimethylamino)ethyl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-1-propanoylpiperidine-3-carboxamide
3-({1-[3-(dimethylsulfamoyl)propyl]pyrrolidin-3-yl}methyl)benzoic acid
4-{2-[1-(4-chloro-2-methoxybenzoyl)piperidin-2-yl]ethyl}morpholine
1-(adamantan-1-yl)-4-(1H-imidazol-2-ylmethyl)piperazine
ethyl 4-(2-amino-4-phenylpyrimidine-5-amido)piperidine-1-carboxylate
2-[4-(1-methoxypropan-2-yl)piperidine-1-carbonyl]-N-(prop-2-en-1-yl)aniline
(2S,4S)-4-[(naphthalen-1-ylmethyl)amino]-1-[(2E)-3-phenylprop-2-en-1-yl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(1-ethyl-1H-imidazol-5-yl)methyl]-1H-1,2,3-triazole
3-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-5-propyl-1,2-oxazole
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine
8-methoxy-2-(1-methyl-1H-pyrazol-4-yl)-3-(1H-pyrazol-1-ylmethyl)quinoline
1-[(2,4-dichlorophenyl)methyl]-3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
2-(ethoxymethyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(hydroxymethyl)-1-[4-(pyrrolidin-1-yl)benzoyl]azepan-4-ol
8-cyclohexyl-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(4-{1-[2-(azepan-1-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)butan-2-ol
2-[methyl(phenyl)amino]-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3,5-dichloro-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-4-methylbenzamide
(4aR,7aS)-1-acetyl-4-[(4-phenylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-ethylpiperidin-2-one
3-(furan-2-yl)-5-{thieno[2,3-d]pyrimidin-4-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[4-(2-chlorophenoxy)piperidin-1-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
4-(3-hydroxy-1,2-oxazole-5-carbonyl)-9-(2-hydroxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[1-(pyrimidin-4-yl)ethyl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide