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1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3,3,3-trifluoropropan-1-one
1-methyl-4-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}piperazine
2-({[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]oxy}methyl)pyridine
[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl][1-(1H-imidazol-1-yl)propan-2-yl]amine
N-methyl-N-{[3-(trifluoromethyl)-1H-pyrazol-5-yl]methyl}oxan-4-amine
7-(2-methoxypyridine-3-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[2-(2-chlorophenyl)ethyl]propanamide
N-[(1-propyl-1H-pyrazol-4-yl)methyl]oxolane-3-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-[2-(2-hydroxyethoxy)ethyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-(pyridin-4-ylsulfanyl)acetamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
8-cyclopropanecarbonyl-2-[(5-methylfuran-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(2,3-dihydro-1H-inden-2-yl)-5-methyl-N-propyl-1,3-oxazole-4-carboxamide
(3aS,6aS)-2-(dimethylcarbamoyl)-5-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentane-1,2-dione
2-[8-(3-methoxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-6-methylpyridine-3-carbonitrile
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazole-3-carboxamide
1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(thian-4-yl)piperazine
1-[(5-chlorothiophen-2-yl)methyl]-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
5-(1-ethyl-1H-imidazol-5-yl)-1-(furan-3-ylmethyl)-4-phenyl-1H-imidazole
4-[3-(2-phenylethyl)piperidin-1-yl]pyrimidin-2-amine
5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
5-{1-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-imidazol-2-yl}-2-(furan-2-yl)pyrimidine
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-(2-methylpyrimidin-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(2-phenoxyethyl)piperidine-3-carboxamide
4-{4-[1-(4-chlorophenyl)cyclopropanecarbonyl]piperazin-1-yl}-2-(3,4-dimethoxyphenyl)-2,3-dihydro-1H-isoindole-1,3-dione
8-(3,5-difluoropyridine-2-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
N-methyl-N-(oxan-2-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl](pyridin-2-yl)methanol
2-[3-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)phenyl]-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-4-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(3-methylphenyl)-1H-pyrazole-4-carboxamide
9-(3-fluorobenzoyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(4-chloro-3-methylphenyl)-2-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]acetamide
4-[3-(ethylcarbamoyl)pyrrolidin-1-yl]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
N-cyclopentyl-5-cyclopropyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1,2-oxazole-3-carboxamide
5-methyl-6-(3-methylpiperidine-1-carbonyl)-N-[2-(piperidin-1-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
5-{4-[4-(3-chlorophenyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-2-methyl-1,4-dihydropyridin-4-one
2-(1-butyl-1H-pyrazol-4-yl)-N,N,6-trimethylquinoline-4-carboxamide
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(2-phenyl-1,3-thiazol-5-yl)methyl]amine
4-(2,3-dihydro-1H-inden-2-yl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-methyl-6-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-4-yl}pyrimidin-4-ol
9-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-1-cyclopentyl-3-(2-methylphenyl)pyrrolidine-2,5-dione
N-(2,3-dimethylphenyl)-3-[(3,4-dimethylphenyl)amino]piperidine-1-carboxamide
{1-[(2-ethoxyphenyl)methyl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-{[2-amino-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]methyl}phenol
(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]{[1-(propan-2-yl)piperidin-4-yl]methyl}amine
2,4-dimethyl-6-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-5H,6H-furo[2,3-d]pyrimidine