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N3-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]piperidine-1,3-dicarboxamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(2-methoxyphenoxy)ethan-1-one
2-butyl-4-{[5-(methoxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(naphthalen-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}ethane-1-sulfonamide
methyl 9-(oxan-2-ylmethoxy)-7-oxo-3-[3-(thiophen-2-yl)propanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-(piperidine-1-carbonyl)piperidine
5-(hydroxymethyl)-2-methyl-4-{[4-(3-methylthiophen-2-yl)-1H-1,2,3-triazol-1-yl]methyl}pyridin-3-ol
1-[(3-fluorophenyl)methyl]-4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-2-one
1-(2-methylpropyl)-2-{1-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-1,2,3-triazol-4-yl}-1H-1,3-benzodiazole
1-(2,3-dihydro-1H-inden-2-yl)-4-[(pyridin-4-ylmethyl)amino]pyrrolidin-2-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}cyclopentanecarboxamide
1-[2-({[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl}amino)ethyl]piperidin-4-ol
1-[4-(2-phenoxyethyl)piperazine-1-carbonyl]isoquinoline
4-(6-methoxypyrimidin-4-yl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(2-chlorophenoxy)-1-(1H-imidazol-2-ylmethyl)piperidine
3-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidine-1-carbonyl)pyridin-2-ol
2-(4-chlorophenyl)-N-phenylmorpholine-4-carboxamide
5-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-methyl-4-phenyl-9-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
8-[2-(2,6-dimethoxyphenoxy)ethyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
5-methanesulfonyl-1'-(3-methyloxetane-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-cyclopropanecarbonyl-2-[3-(furan-2-yl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[1-(2-methoxyphenyl)-1H-imidazol-2-yl]-1-methylpiperidine
N-(1H-imidazol-2-ylmethyl)-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
5,5-diphenyl-1-[1-(pyrazin-2-yl)propan-2-yl]piperidin-2-one
(4aR,7aS)-1-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{methyl[4-(methylamino)pyrimidin-2-yl]amino}-1-phenylpropan-1-ol
(3aS,6aS)-2-(ethanesulfonyl)-5-(3-phenylpropyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-{[(quinoxalin-2-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
2,2-dimethyl-N-{5-methyl-3-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]thiophen-2-yl}propanamide
3-methoxy-1-[4-(2-methylphenoxy)piperidin-1-yl]propan-1-one
8-chloro-2-{[4-(4-methylpyrimidin-2-yl)piperazin-1-yl]methyl}quinoline
5-methyl-N-{[1-(phenoxymethyl)cyclopropyl]methyl}pyrimidin-2-amine
2-(1-methyl-1H-pyrazol-4-yl)-4-[4-(pyridin-2-yl)piperazine-1-carbonyl]quinoline
1-(azepan-1-yl)-3-[3-({[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
4-[3-(3-chlorophenyl)-3-phenylpropanamido]-N,N-dimethylbutanamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-ethylpyrimidine-5-carboxamide
3-(4-hydroxyphenyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}benzamide
1-{1-[4-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-3-yl}pyrrolidin-2-one
6-cyano-N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyridine-3-carboxamide
3-[(4-ethylpiperazin-1-yl)methyl]-2-(3-methoxyphenyl)-7-(methylsulfanyl)quinoline
2-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-4-(propan-2-yl)-1,3-thiazole
3-methoxy-5-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzoic acid
(4aS,8aR)-6-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
2-(1-propylpiperidin-4-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]acetamide
2-methyl-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]imidazo[1,2-a]pyrimidine-3-carboxamide
1-(azocan-1-yl)-3-(2-methoxy-5-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
3-({[(2-fluorophenyl)methyl](2-methoxyethyl)amino}methyl)-6-methyl-4H-chromen-4-one
(4aS,7aR)-1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-benzyl-3-ethyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1,4-diazepan-5-one