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2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(2-hydroxyethyl)-N-(propan-2-yl)acetamide
2-(3-{3-[cyclohexyl(methyl)amino]propyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)-N-methylacetamide
8-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[(2E)-4-methylpent-2-en-1-yl]piperidin-3-ol
1-[1-(3-cyclohexylpropanoyl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(2-methoxyethyl)-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine-3-carboxylic acid
3-butyl-1-(4-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}phenyl)urea
N-{[6,7-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)thiophene-2-carboxamide
1-(4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)butan-1-ol
(1R,6S)-9-methyl-3-{[5-(pyridin-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
N-cyclooctyl-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
1-[3-(5-methyl-2-{[2-(morpholin-4-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]-2-(2,3,6-trifluorophenyl)ethan-1-one
1-[2-(dimethylamino)ethyl]-4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amine
N-[1-(2-ethylbutyl)piperidin-4-yl]methanesulfonamide
1-(4-acetylphenyl)-3-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]urea
N-(3,3-dimethyl-2-oxobutyl)-4-(quinolin-6-yloxy)piperidine-4-carboxamide
4-(3-methylpyridin-4-yl)-N-[3-(1H-1,2,4-triazol-1-yl)phenyl]-1,4-diazepane-1-carboxamide
2-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-2,7-diazaspiro[4.5]decane
8-(1H-imidazol-4-ylmethyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
[3-(2-methoxyethyl)-1-[3-(methylsulfanyl)propyl]piperidin-3-yl]methanol
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(2-methyl-1H-indol-1-yl)propanamide
N-[1-(methoxymethyl)cyclopentyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-[4-(adamantan-2-yl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[4-(3-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(1,7-dimethyl-1H-indole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-methyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyrimidin-2-amine
(1R,5S,6R)-3-(1-phenylcyclohexanecarbonyl)-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
5-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-5-oxopentanamide
N,N-dimethyl-2-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]aniline
(4aR,7aS)-1-(2-methylpropanoyl)-4-(3-phenylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[3-cyclopropyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
4-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}-1-{spiro[2.3]hexane-1-carbonyl}piperidine
N-(1-methyl-1H-1,2,4-triazol-3-yl)-3-({methyl[1-(pyridin-2-yl)propan-2-yl]amino}methyl)benzamide
(3R,5S)-N3-(4-fluorophenyl)-N5-(2-methylpropyl)piperidine-3,5-dicarboxamide
4-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)methyl]-2-methoxyphenol
2-(4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperazin-1-yl)pyrazine
5-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]pyrrolidin-2-yl}-N-(1-methyl-1H-pyrazol-4-yl)thiophene-2-carboxamide
2-(4-hydroxyphenyl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
1-[(2-fluorophenyl)methyl]-6-oxo-N-[3-(pyridin-2-yl)propyl]piperidine-3-carboxamide
1-[4-(1H-imidazol-1-yl)phenyl]-N-[(2R)-3-methylbutan-2-yl]piperidin-4-amine
N-[(2S,3S)-1-hydroxy-3-methylpentan-2-yl]-3-(2-methyl-1H-indol-1-yl)propanamide
1-[1-(2-hydroxyacetyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
2-(2-methoxybutanoyl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
2-(1-ethyl-1H-imidazol-5-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
(5-{4-phenyl-1-[1-(pyridin-3-yl)propyl]-1H-imidazol-5-yl}furan-2-yl)methanol