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methyl (2S)-2-{[1-cyclohexyl-5-(cyclopropylcarbamoyl)-4-oxo-1,4-dihydropyridin-3-yl]formamido}-2-phenylacetate
2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[4-(pyridin-2-yl)butyl]acetamide
3-(2-hydroxyethyl)-4-{2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}piperazin-2-one
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
1-methyl-N-(pyridin-4-ylmethyl)-5-[(2,2,2-trifluoroethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[4-methyl-6-(pyrrolidine-1-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]-1-(morpholin-4-yl)ethan-1-one
1-{1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](oxolan-2-ylmethyl)amine
N-{3-[4-hydroxy-4-(hydroxymethyl)azepane-1-carbonyl]-4,5-dimethylthiophen-2-yl}-2-methylpropanamide
1-{2-[4-(difluoromethoxy)phenyl]-1H-imidazol-1-yl}butan-2-ol
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-3-(methoxymethyl)pyrrolidine
2-(2-{[2-methoxy-2-(thiophen-2-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
(1S,6R)-9-[(1-phenyl-1H-pyrazol-5-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
9-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-2-[3-(dimethylamino)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
7-methyl-4-(4-methylpiperidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
(2R)-3-methyl-2-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)butanamide
1-{2-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-benzyl-5-[5-(methoxymethyl)furan-2-yl]-1H-1,2,4-triazole
3-(2-{6-azabicyclo[3.2.1]octan-6-yl}-2-oxoethyl)-1-[2-(dimethylamino)ethyl]-3-(2-methylphenyl)pyrrolidine-2,5-dione
(2S)-2-[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]butan-1-ol
(2S)-2-cyclohexyl-2-{[3-(4-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}acetic acid
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
6-fluoro-2-oxo-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
5-(2-methoxy-4-methylphenoxymethyl)-N-[(2S)-oxolan-2-ylmethyl]-1,2-oxazole-3-carboxamide
2-(3-methoxyphenyl)-N-(oxan-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
3-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
1-cyclopropyl-N-[(3,4-difluorophenyl)methyl]-1H-pyrrole-2-carboxamide
3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-1-(3,5-dimethyl-1H-pyrazole-4-carbonyl)piperidine
(5S,9aS,9bS)-5-[4-(benzyloxy)phenyl]-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3R,4R)-3-cyclopropyl-1-(2,3-difluoro-6-methoxybenzoyl)-4-methylpyrrolidin-3-ol
N-{[(2S,4S)-1-[(5-chlorothiophen-2-yl)sulfonyl]-4-fluoropyrrolidin-2-yl]methyl}propanamide
9-(2-amino-5-ethyl-6-methylpyrimidin-4-yl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-[2-(oxan-4-yl)ethyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-[3-(furan-2-yl)-1H-pyrazol-5-yl]piperidine
1-[4-(1H-pyrazol-3-yl)benzoyl]azocane
2-[1-(1-methylpiperidin-4-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
2-methyl-1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
N-(4-fluoro-2-methylphenyl)-3-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)propanamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}acetamide
2-(1,7-dimethyl-1H-indole-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridazine
5-[1-benzyl-5-(dimethylamino)-1H-1,2,4-triazol-3-yl]pyridin-3-amine
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-(2,2,2-trifluoroethyl)piperazine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(dimethylamino)butan-2-yl]-1,3-oxazole-4-carboxamide
1-(6-chloro-1,3-benzothiazol-2-yl)-N-[3-(1H-imidazol-2-yl)propyl]piperidin-4-amine
2-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}benzonitrile
N-[(3,4-difluorophenyl)methyl]-1-(methoxymethyl)cyclopropane-1-carboxamide