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5-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-N-methylpyrimidin-2-amine
(3aR,5S,6S,7aS)-2-[(5-phenylthiophen-2-yl)methyl]-octahydro-1H-isoindole-5,6-diol
4-[3-(2-cyclopentyl-1H-imidazol-1-yl)propyl]morpholine
4-(5-methyl-1,2,4-oxadiazol-3-yl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]acetamide
(2R,3R,6R)-3-phenyl-5-(pyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1s,4s)-4-[2-(3-fluoro-2,4-dimethylphenyl)-1H-imidazol-1-yl]cyclohexan-1-amine
1-(6-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}pyridin-3-yl)ethan-1-one
1-{6-[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]pyridin-3-yl}ethan-1-one
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)piperidin-2-one
2-(3-methoxypropyl)-1-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]piperidine
2-(1-methyl-1H-imidazol-2-yl)-1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
N-({5-[(3-ethoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
N-(1-benzothiophen-2-ylmethyl)-N,5-dimethyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
ethyl 4-({2-[(4-fluorophenyl)methyl]morpholin-4-yl}methyl)-1H-pyrazole-3-carboxylate
6-chloro-N-[2-(pyrrolidine-1-sulfonyl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
(2S)-3-(1H-imidazol-4-yl)-2-{4-[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]-1H-1,2,3-triazol-1-yl}propanoic acid
1-[ethyl(methyl)sulfamoyl]-4-phenoxypiperidine-4-carboxylic acid
4-[4-({[(2S)-1-ethylpyrrolidin-2-yl]methyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
2-(ethylamino)-4-methyl-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1,3-thiazole-5-carboxamide
2-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
[(3,7-dimethyl-1H-indol-2-yl)methyl](methyl)(pyridin-2-ylmethyl)amine
4-[4-(1H-pyrazol-5-yl)phenyl]-5H,6H,7H-cyclopenta[d]pyrimidin-2-amine
6-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
1-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
1-(3,5-dimethylphenyl)-4-(5-fluoropyridin-2-yl)piperazin-2-one
6-chloro-N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)imidazo[1,2-a]pyridine-2-carboxamide
5-(1H-indol-1-ylmethyl)-N-(2-oxopiperidin-3-yl)-1H-pyrazole-3-carboxamide
methyl 3-{[1-(cyclopropylmethyl)-5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
1-{3-[5-(4-fluoro-2-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
methyl[(3-methyl-1,2-oxazol-5-yl)methyl][(1-propyl-1H-imidazol-2-yl)methyl]amine
1-[(5-{[3-(2-hydroxyethoxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]-3,3-dimethylurea
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[4-(pyridin-3-ylmethyl)piperazin-1-yl]propan-1-one
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]acetamide
[(2-chloro-4-fluorophenyl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N-[2-methyl-2-(morpholin-4-yl)propyl]-5-(propan-2-yl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
5-ethyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}pyrimidin-2-amine
2-tert-butyl-6-(4-fluoro-3-methylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-{2-[4-(4-chlorophenyl)-4H-1,2,4-triazol-3-yl]ethyl}phenol
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)prop-2-ene-1-sulfonamide
N-[2-(2-fluorophenyl)ethyl]-5-{1-[(2-fluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-1-benzofuran-2-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}acetamide
N-[2-fluoro-5-(trifluoromethyl)phenyl]-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
1-ethyl-4-{[2-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-imidazol-1-yl]methyl}-5-methyl-1H-pyrazole
5-[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]-1-[(2-methylphenyl)methyl]azepan-2-one
2-[(6-ethoxypyridin-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
5-fluoro-1-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazole
3-[(4-fluorophenyl)formamido]-N-{3-[(pyridin-3-yl)amino]propyl}propanamide