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5-acetyl-N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[3-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethoxy)phenyl]propanamide
4-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2-methoxypyridine-3-carbonitrile
2-hydroxy-5-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}benzoic acid
6-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-oxo-4-phenyl-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-(cyclobutylmethyl)-5-(2-phenylethyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
1-(2-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}ethyl)-4-(pyridine-4-carbonyl)piperazine
6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-N,N-dimethylpyrazin-2-amine
2-{[(3-hydroxypropyl)(pyridin-4-ylmethyl)amino]methyl}-6,8-dimethylquinolin-4-ol
5-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
4-({[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)benzene-1-sulfonamide
3-(oxolan-2-ylmethyl)-5-[3-(1H-pyrazol-4-yl)phenyl]-1,2,4-oxadiazole
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)ethan-1-one
N-(5-cyanopyridin-2-yl)-4-{[4-(prop-2-en-1-yl)piperazin-1-yl]methyl}benzamide
4-{3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanoyl}-1λ6-thiomorpholine-1,1-dione
4-(2-methoxyphenoxy)-1-(pyrrolidin-3-ylmethyl)piperidine
3-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-2-methylthieno[3,2-d]pyrimidin-4-amine
1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-[4-ethyl-5-oxo-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(pyrazin-2-yl)acetamide
(2-{1-[(5-chlorofuran-2-yl)methyl]piperidin-2-yl}ethyl)dimethylamine
6-{3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
methyl 6-(2,2-diphenylacetyl)-2-(methylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{4-[(2-chlorophenyl)methyl]-3-oxo-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl}-1,4-diazepane-1-carbaldehyde
5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-one
N-[(5,6-dimethylpyridin-3-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-[1-(cyclohex-1-en-1-yl)ethyl]-3-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]urea
(2S)-3-(4-hydroxyphenyl)-2-{[6-(methoxymethyl)pyrimidin-4-yl]amino}propanamide
1-(3-{[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}piperidin-1-yl)ethan-1-one
[(5-tert-butyl-1H-pyrazol-3-yl)methyl][2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]methylamine
4-[(1R)-1-(4-fluorophenyl)ethyl]-3-(3-hydroxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(2,2-diphenylacetyl)-1,4-diazepan-5-one
3-{[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}pyrrolidin-3-ol
1-{[2-(1H-imidazol-1-yl)phenyl]methyl}-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
1-(benzyloxy)-3-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propan-2-ol
N-(2-methoxyethyl)-N-methyl-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl][1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
3-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-3-[methyl({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})amino]propanamide
2-(1H-indol-3-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethan-1-one
2-{[(3,5-dimethylphenyl)methyl]sulfanyl}-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]acetamide
3-[2-(3,5-dimethoxyphenyl)acetyl]-3,9-diazaspiro[5.6]dodecan-10-one
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-propylpiperidine-3-carboxylic acid
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[1-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
2-(1-{3-[(1-methylpiperidin-4-yl)oxy]propyl}-1H-imidazol-2-yl)benzoic acid
1-ethyl-6,7,8-trifluoro-N-methyl-4-oxo-N-(pentan-3-yl)-1,4-dihydroquinoline-3-carboxamide
4-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}-N-(1,2,3-thiadiazol-5-yl)benzamide
9-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-{2-[1-(1H-imidazole-2-carbonyl)piperidin-2-yl]ethyl}phenol
(2S,4S)-N-ethyl-1-[(5-methylfuran-2-yl)methyl]-4-[2-(morpholin-4-yl)acetamido]pyrrolidine-2-carboxamide