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3-[(3R,4S)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-{1-[3-(methylsulfanyl)butyl]piperidin-4-yl}-1H-1,3-benzodiazole
(1S,5R)-6-(cyclopropylmethyl)-3-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(diphenylmethyl)-N-methyl-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
8-fluoro-2-[4-(2-oxopyrrolidin-1-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
2-[(3-methoxyphenyl)amino]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]butanamide
(3R,4S)-1-{2-[2-(3-methoxyphenyl)ethyl]benzoyl}-4-propylpyrrolidin-3-amine
2-(methylsulfanyl)-5-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}pyrimidine
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-cyclopropyl-2-methoxybenzamide
N-benzyl{[2-(2-hydroxyethyl)phenyl]amino}sulfonamide
1-benzyl-8-[(9-ethyl-9H-carbazol-3-yl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(6-methylpyridazin-3-yl)piperidin-3-ol
4-(1-tert-butyl-1H-pyrrole-3-carbonyl)-1-(cyclopropylmethyl)-2-(propan-2-yl)-1,4-diazepane
3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
4-(hydroxymethyl)-1-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]piperidin-4-ol
4-[(4-methylphenyl)methyl]-11-[(1,2-oxazol-3-ylmethyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(5S,9aS,9bS)-5-(1-benzothiophen-2-yl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-acetyl-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
6-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyrimidin-4-amine
(1R,5R)-6-(naphthalen-1-ylmethyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3-hydroxy-1,2-oxazol-5-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylpropanamide
N2-(2,2-dimethylpyrrolidin-3-yl)-N1-(pyridin-3-yl)ethane-1,2-diamine
(3R,4R)-1-(cyclohex-1-ene-1-carbonyl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
1-{[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]amino}-3-phenylpropan-2-ol
2-(5-amino-1,3,4-thiadiazol-2-yl)-N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}acetamide
8-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl 3-benzamido-5-{[(2,6-dimethoxyphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(2-oxopyrrolidin-1-yl)benzamide
5-[4-(benzyloxy)butyl]pyridin-3-amine
5-[5-(piperazin-1-ylmethyl)thiophen-3-yl]pyrimidine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)cyclobutanamine
5-(3,4-dimethoxyphenyl)-N-methyl-N-[4-(morpholin-4-yl)butyl]-1,2,4-triazin-3-amine
1-{2-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}thiophene-2-carboxamide
(3aS,6aR)-5-(2-hydroxypyridine-3-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-N-(furan-2-ylmethyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
5-acetyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]thiophene-2-carboxamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
1-(4-fluorophenyl)-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-3-(methoxymethyl)piperidine
7-(4-amino-5-methylpyrimidin-2-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5,6-dimethylpyrimidine
N,N,5,7-tetramethyl-2-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
4,6-dimethyl-2-oxo-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(4-fluorophenoxymethyl)-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(1H-pyrazole-4-carbonyl)piperidine
3-{4-[(2,3-dichloro-4-methylphenyl)methyl]piperazin-1-yl}pyrazine-2-carbonitrile
2-(4-fluorophenyl)-1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)azetidine
2-[(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]acetic acid