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3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-1-[2-(4-fluorophenyl)pyrrolidin-1-yl]propan-1-one
N-{1-[4-(3-chlorophenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-2,6-dimethoxybenzamide
1'-(3-hydroxypyridine-2-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N,5-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrazine-2-carboxamide
methyl 2-[(prop-2-en-1-yl)sulfamoyl]-6-[3-(trifluoromethyl)benzoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,2-oxazole-3-carbonyl)piperidine
(4aR,7aS)-1-[2-(azocan-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}morpholine
N-cyclopropyl-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}propanamide
N-methyl-5-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
[1-({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)azepan-2-yl]methanol
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})(oxolan-2-ylmethyl)amine
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(5-propylthiophene-3-carbonyl)-1,4-diazepan-5-one
1-cyclobutanecarbonyl-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-methylacetamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylpyridin-2-yl)methyl]amine
3-{1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-4-{[(2,5-difluorophenyl)methyl]amino}-1-[(2E)-3-phenylprop-2-en-1-yl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(1H-pyrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
4-({1-ethyl-5-[2-(1H-1,2,4-triazol-1-yl)phenyl]-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine
3-{2-[(4-cyclopentylpyrimidin-2-yl)amino]-1-hydroxyethyl}phenol
1-methyl-4-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{2-hydroxy-3-[2-methoxy-4-({[2-(3-methoxyphenyl)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
2-(dimethyl-1,2-oxazol-4-yl)-N-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}pyrrolidine-1-carboxamide
3-[1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]-4-methoxybenzene-1-sulfonamide
N-[2-(dimethylamino)ethyl]-1-[1-(2-phenylpropyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
3-[1-(4-chloro-2-fluorobenzoyl)piperidin-3-yl]benzoic acid
3-{methyl[2-(pyridin-2-yl)ethyl]amino}-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide
[(2S)-1-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)pyrrolidin-2-yl]methanol
(2S)-5-carbamimidamido-2-({6-methylimidazo[1,2-a]pyridin-2-yl}formamido)pentanoic acid
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-[3-(methylsulfanyl)phenyl]ethan-1-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(pyridin-4-yl)acetamide
3-(2-methyl-1H-indol-1-yl)-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide
6-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2,3,4-tetrahydroquinoline
6-(4-fluorophenyl)-N-[(1-hydroxycyclohexyl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(butan-2-yl)-3-(1H-imidazol-2-yl)-N-[(3-methylthiophen-2-yl)methyl]benzamide
2-[(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)methyl]benzonitrile
1-{4-[2-(naphthalen-1-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}-2-phenylethane-1,2-dione
2-[3-(1H-indol-3-yl)-5-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-1,2,4-triazol-1-yl]acetic acid
(1-benzothiophen-2-ylmethyl)(methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
4-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydroquinolin-2-one
3-{1-[2-(2,3-dimethylphenoxy)acetyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-cyclopentyl-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyrimidin-2-amine
2-methyl-N-(2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)propanamide
N-cyclopropyl-N-[1-(pyrimidin-4-yl)piperidin-4-yl]benzenesulfonamide
ethyl 4-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}piperidine-1-carboxylate