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(4aR,7aS)-1-[2-(3,3-diethylpyrrolidin-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-4-methylpiperazine
2-(2-{1-[2-(1,2-benzoxazol-3-yl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-(pyrimidin-4-ylmethyl)acetamide
(5S,9aS,9bS)-5-(1-benzofuran-2-yl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-{[2-(4-hydroxyphenyl)ethyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-amino-4-(4-hydroxy-3,5-dimethoxyphenyl)-5H,6H,7H,8H,9H,10H-cycloocta[b]pyridine-3-carbonitrile
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(5-hydroxypyrazine-2-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
{1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]azepan-2-yl}methanol
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(dimethylamino)benzamide
2-(2-{1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
6-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-5,6-dihydro-1,6-naphthyridin-5-one
5-[3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]pyrazin-2-ol
methyl (1R,3S,3aR,6aS)-5-ethyl-3-(furan-3-yl)-1-(2-methoxy-2-oxoethyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[3-(2-propoxyphenyl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[3-(pyridin-2-yl)propyl]pyrimidine-5-carboxamide
3-[(3S,4S)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
1-[benzyl(methyl)amino]-3-(4-{[(oxan-4-ylmethyl)amino]methyl}phenoxy)propan-2-ol
{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
4-(3,3-difluoropiperidine-1-carbonyl)-7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
3-(4-fluorophenyl)-4-(1-propyl-1H-pyrazole-5-carbonyl)piperazin-2-one
N-(2-methylpropyl)-2-(methylsulfanyl)-N-(pyridin-2-ylmethyl)pyridine-3-carboxamide
6-(methoxymethyl)-N,1-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(3,4-difluorophenyl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
2-cyclopropyl-4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]quinoline
2-(ethylamino)-N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}pyrimidine-5-carboxamide
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1H-1,2,3-benzotriazole-5-carboxamide
3-(hydroxymethyl)-N-[2-(prop-2-en-1-yloxy)phenyl]piperidine-1-carboxamide
N-[(2R,3R)-1'-(3-cyclohexylpropanoyl)-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]cyclopropanecarboxamide
1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-4-(pyrrolidine-1-carbonyl)piperidine
N-[(1-{[2-(difluoromethoxy)phenyl]methyl}pyrrolidin-3-yl)methyl]cyclobutanecarboxamide
N-(1,1-dioxo-1λ6-thian-4-yl)-6-fluoro-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(phenylsulfanyl)acetamide
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-5-(hydroxymethyl)furan-2-carboxamide
1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}-2-(pyridin-2-yl)ethan-1-one
6-(1-benzothiophen-2-ylmethyl)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
3-{2-[4-(morpholine-4-carbonyl)piperazin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
7-(cyclopropylmethyl)-2-{[2-(difluoromethoxy)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(1H-pyrazol-1-yl)butanamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(5-methyl-1,3-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[3-({[(1R)-1-(3-methoxyphenyl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
8-(5-methylpyridin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}phenoxy)ethan-1-ol
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
N-[1-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]pyrimidin-2-amine
1-(3-benzoylpiperidin-1-yl)-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
1-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(1H-pyrazol-3-yl)piperidine