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N-methyl-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]benzonitrile
3-(1H-imidazol-2-yl)-N-[1-(2-methylphenyl)cyclopropyl]benzamide
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-(2,2,2-trifluoroethyl)acetamide
4-hydroxy-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
2-({2,6-dimethylimidazo[1,2-a]pyridin-3-yl}formamido)-N-(2-fluoro-4-methylphenyl)acetamide
2-(6-hydroxy-4-propyl-1,4-diazepan-1-yl)-N-(pyridin-2-ylmethyl)acetamide
(4-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
2-{[2-oxo-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]methyl}benzonitrile
1-cyclopropyl-N-[(3S,5S)-5-(diethylcarbamoyl)-1-propanoylpyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
3-(methanesulfonylmethyl)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidine
4-[4-(4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]-1-(3-methylbutyl)piperidine
(2S,4S)-4-amino-1-{[5-(4-chlorophenoxy)-1,3-dimethyl-1H-pyrazol-4-yl]methyl}-N-methylpyrrolidine-2-carboxamide
1-[(1S,5R)-6-(4-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
(3aS,6aS)-5-(8-methoxyquinolin-2-yl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}ethyl)pyrrolidin-2-one
1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}piperidin-3-ol
5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-N-[1-(thiophen-2-yl)propyl]-1H-1,3-benzodiazole-7-carboxamide
[1-(2-amino-6-methoxypyrimidin-4-yl)-3-ethylpiperidin-3-yl]methanol
N-(2,4-dimethylphenyl)-2-oxo-2-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}acetamide
(6-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}pyridin-2-yl)methanol
N-{2-[1-({5-[(N-methylmethanesulfonamido)methyl]furan-2-yl}methyl)piperidin-2-yl]ethyl}acetamide
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-6-methyl-2-oxo-4-(thiophen-2-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(1H-imidazol-1-yl)ethyl]piperidine-3-carboxamide
1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-(2-methyl-1H-imidazol-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
2-[2-(4-chlorophenyl)morpholin-4-yl]-5-methylpyrimidin-4-amine
1-(carbamoylmethyl)-N-{1-[(3-chlorophenyl)amino]-2-methylpropan-2-yl}piperidine-3-carboxamide
2-{[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}benzoic acid
1-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2-{1-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
4-[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazine-1-carbonyl]phenol
6-(4-hydroxy-3,5-dimethoxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
2-cyclopropanecarbonyl-8-(6-ethyl-2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,5R)-6-(3,5-dimethoxybenzoyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
9-methyl-2-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-[(3-fluorophenyl)methyl]piperazine
2-(furan-2-yl)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]azepane
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-(1,3-thiazol-5-yl)ethan-1-one
N-(1,3-dihydroxy-2-methylpropan-2-yl)-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
5-methyl-1-(2-methylphenyl)-4-[2-(1-propylpiperidin-4-yl)acetyl]piperazin-2-one
1-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-1-(4-methylpyrimidin-2-yl)piperidin-4-amine
2-(2-phenylethyl)-8-(thiophen-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-benzyl-N-[2-(dimethylamino)ethyl]-2-methylpyrimidine-5-carboxamide
1-[(4-chlorophenyl)methyl]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide