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1-{2-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydroquinolin-2-one
2-{1-[(5-methylfuran-2-yl)methyl]-4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl}ethan-1-ol
(2-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-oxoethyl)urea
2-[(1S,5R)-3-(2,6-difluorobenzoyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-[(3-chlorophenyl)methyl]-4-{4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-(2-fluorophenyl)ethyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
N-{5-methoxy-2-[(2S)-2-methoxy-2-phenylacetamido]phenyl}-2-methylpropanamide
2-(3-methoxypropyl)-8-(pyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-3,3-dimethylbutan-1-one
3-(dimethylamino)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
7-(3-chlorophenyl)-4-(4-methyl-1,3-oxazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{1-[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]piperidin-3-yl}propan-1-one
methyl (2S)-1-(2-{4-[4-({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)piperidin-1-yl]phenyl}acetyl)pyrrolidine-2-carboxylate
5-{[(2-chloropyridin-3-yl)methyl](methyl)amino}-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)-4-(pyridin-3-yl)pyrimidin-2-amine
3-(1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
1-(2-methoxyethyl)-3,8-bis(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}benzamide
N-cyclopentyl-2-{ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}propanamide
3-(3,4-difluorophenyl)-5-[(1R,2S)-2-propylcyclopropanecarbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[1-(2-hydroxyethyl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]-1-(3-hydroxyphenyl)pyrrolidin-2-one
N-[1-(2,5-difluorophenyl)cyclopropyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
3-(2-methoxyphenyl)-1-(3-methoxypropyl)-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
{1-[2-(benzenesulfonyl)ethyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
4-(4-methyl-1H-pyrazol-1-yl)-1-[(2S)-1-(propan-2-yl)pyrrolidine-2-carbonyl]piperidine-4-carboxylic acid
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(1-cyclohexyl-1H-pyrazol-5-yl)-1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
8-(1H-imidazol-2-ylmethyl)-1-(2-methoxyethyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
methyl 5-{[(4-chlorophenyl)methyl]amino}-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-methyl-4-{1-[2-(1H-pyrazol-4-yl)ethyl]piperidin-3-yl}-6-(pyrrolidin-1-yl)pyrimidine
3-[benzyl({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amino]propanamide
2-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)pyrazine
2-ethyl-4-[2-(3-fluorophenyl)piperidine-1-carbonyl]pyridine
N2-(2,2-dimethylpyrrolidin-3-yl)-N1-(4-methylpyridin-2-yl)ethane-1,2-diamine
2-(morpholin-4-yl)-2-(thianthren-1-yl)acetic acid
N-ethyl-2-(4-oxocyclohexyl)-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}acetamide
3-(3-fluorophenyl)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
1-[(5-chlorothiophen-2-yl)methyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-[2-(1H-imidazol-2-yl)benzoyl]-4-[(2-methylphenyl)sulfanyl]piperidine
3-[(2-fluorophenyl)formamido]-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}propanamide
4-(4-cyclohexanecarbonylpiperazine-1-carbonyl)-7-fluoro-2-methylquinoline
1-{2-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]ethyl}pyrrolidin-2-one
2-{3-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)formamido]propanamido}acetic acid
1'-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one