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N'1-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopropane-1,1-dicarboxamide
8-[(2R,3S)-2-amino-3-hydroxybutanoyl]-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
6-methoxy-N-methyl-2-oxo-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-{6-[3-(1H-pyrazol-3-yl)phenyl]-1,2,3,4-tetrahydroquinolin-1-yl}ethan-1-one
4-(3-fluorophenoxy)-1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}piperidine-4-carboxylic acid
2-methyl-6-(1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperidin-4-yl)pyrimidin-4-ol
4-[2-(4,5-diphenyl-1H-imidazol-1-yl)ethyl]pyridine
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N,6-dimethylpyrimidin-4-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)propanamide
1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
(4aS,7aR)-1-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2-fluorophenoxy)-1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperidine
N-(3-hydroxypropyl)-1-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]azepane-2-carboxamide
1-[3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanoyl]-N-(1-methoxypropan-2-yl)piperidine-4-carboxamide
1-(4-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)ethan-1-one
2-(4-methoxyphenyl)-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(2S,4S,5R)-1,2-dimethyl-5-phenyl-4-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]pyrrolidine-2-carboxylic acid
4-[8-methyl-3-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)imidazo[1,2-a]pyridine-2-carbonyl]morpholine
3-[({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)methyl]-1λ6-thiolane-1,1-dione
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)(3-methylbutyl)amine
2-chloro-N-(2-{[5-(pyrrolidin-1-ylmethyl)furan-2-yl]formamido}ethyl)benzamide
1-(2-methoxyethyl)-N-{5-[2-(4-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}pyrrolidine-3-carboxamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-[(3-methylphenyl)sulfanyl]piperidine
3-cyclohexyl-N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
1-(cyclohexylmethyl)-3-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}urea
3-(3-chlorophenoxymethyl)-1-methyl-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazole
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
8-[2-(1,1-dioxo-1λ6-thian-4-yl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(5-methylfuran-2-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
N-(2,3-dihydroxypropyl)-5-(3-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
4-[(2,2-difluoroethyl)sulfamoyl]-N-(piperidin-4-ylmethyl)benzamide
(3S,9aR)-2-methyl-3-(2-methylpropyl)-8-(naphthalene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(3-acetyl-1H-indol-1-yl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]butanamide
2-[2-oxo-4-(quinolin-4-ylmethyl)piperazin-1-yl]benzonitrile
4-{[5-(1,2-dihydroacenaphthylen-5-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
1-[4-(5-methyl-1,3-diphenyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]ethan-1-one
[(2-chloro-6-fluorophenyl)methyl](methyl)(pyrazin-2-ylmethyl)amine
methyl(1,3-thiazol-2-ylmethyl){[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
N-(4-methoxy-2-methylphenyl)-3-[1-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)piperidin-3-yl]propanamide
1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
N-(3-cyclopentylpropyl)-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-[3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
4-(4-ethyl-1H-pyrazol-5-yl)piperidine
3-[4-(4-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
methyl (1R,5S,6R)-6-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane-3-carboxylate
5-[1-cyclohexyl-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]-1-methylpiperidin-2-one
methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl][(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
2,6-dimethoxy-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}pyrimidin-4-amine
2-(4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-ol
(1-methyl-1H-imidazol-2-yl)[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]methanol