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1,5-dimethyl-4-[1-(2-methylprop-2-en-1-yl)-4-phenyl-1H-imidazol-5-yl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
dimethyl({4-methyl-5-[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
ethyl 1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(3-phenylpropyl)piperidine-4-carboxylate
1-methyl-4-({5-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
2-amino-6-(4-hydroxyphenyl)-4-(1H-imidazol-4-yl)-5-methylpyridine-3-carbonitrile
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-pentanamidobenzamide
3-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}phenol
3-fluoro-N-(1-phenylbutyl)pyridine-4-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(3-phenoxyphenyl)methyl]acetamide
2-cyclohexyl-6-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-1,3-benzoxazole
N-[2-(pyridin-3-yloxy)propyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
5-chloro-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-methyl-5-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]benzene-1,3-diol
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-(pyridin-3-yl)propan-1-one
6-(2,5-dimethylfuran-3-yl)-2-(3-hydroxyazetidine-1-carbonyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyrrolidin-1-yl)ethane-1,2-dione
5-[4-(3-propoxyphenyl)-1H-pyrazol-1-yl]-1H-1,2,3,4-tetrazole
9-(4-methyl-1,3-thiazole-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-{1-[(2-chlorophenyl)methyl]-1H-imidazol-2-yl}-2-(methoxymethyl)pyrimidine
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-cyclohexylurea
(1S,5R)-6-(1-methyl-1H-pyrrole-2-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[5-(2-acetamidopropyl)-3-ethyl-1H-1,2,4-triazol-1-yl]acetic acid
N-(2-methoxyethyl)-1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
2-methyl-N-(2-oxoazepan-3-yl)-1-benzofuran-5-carboxamide
2-phenyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
N-(6-phenoxypyridin-3-yl)-1-(pyridin-4-ylmethyl)piperidine-2-carboxamide
2-(1H-indazol-1-yl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
3-({1-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]pyrrolidin-3-yl}methyl)benzamide
2-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]-4,6-dimethylpyridine-3-carbonitrile
(1S,4R)-4,7,7-trimethyl-3-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-oxabicyclo[2.2.1]heptane-1-carboxamide
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
(4aS,8aR)-6-[(2E)-hex-2-en-1-yl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
4-ethyl-1-methyl-3-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-cyclopentyl-N-[(4-methanesulfonylmorpholin-2-yl)methyl]propanamide
2-methoxy-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-(pyrimidin-4-ylmethyl)piperidine-3-carboxamide
6-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1,2-dihydropyridin-2-one
N-(1-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
(2S,4R)-N-[2-(2-fluorophenyl)ethyl]-4-{[(4-fluorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}methyl)-3-methylbut-2-enamide
N-[(5-methoxy-1H-indol-2-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
2-{[2-(3-fluorophenoxy)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-[2-(4-phenylpyrimidin-2-yl)ethyl]urea
N-(adamantan-2-yl)-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carboxamide
3-[2-(diethylamino)ethyl]-3-methyl-1-[3-(pyridin-3-yl)phenyl]urea
2-({2-amino-6-[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
2,6-dimethyl-3-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
4-ethyl-6-(4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperazin-1-yl)pyrimidine
N-[(3R,5S)-1-benzyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-2-hydroxypyridine-3-carboxamide