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3-(1H-1,3-benzodiazol-1-yl)-1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propan-1-one
{[3-(3-fluorophenyl)oxolan-3-yl]methyl}[(3-methoxyphenyl)methyl]amine
4-(azepane-1-carbonyl)-7-fluoro-2-methylquinoline
2-(5-chloro-6-hydroxy-2-methylpyrimidin-4-yl)-N,N-bis(propan-2-yl)benzamide
N-butyl-1-[1,3-dioxo-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
(4aS,8aS)-2-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-decahydroisoquinolin-4a-ol
(1S,5R)-6-(cyclobutylmethyl)-3-[3-(4-hydroxyphenyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(dimethylamino)ethyl]-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-1,3-oxazole-4-carboxamide
[(1-methyl-1H-imidazol-2-yl)methyl]({[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(propan-2-yl)amine
1-(1-{4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}ethyl)piperidine
8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentan-1-one
N-(2-hydroxyethyl)-N-methyl-1-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
2-(1,2-benzoxazol-3-yl)-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)acetamide
6-methoxy-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
methyl 9-(oxan-2-ylmethoxy)-7-oxo-3-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[3-(1H-imidazol-1-yl)propyl]acetamide
N-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-ethylphenyl]acetamide
1-[(3S,4R)-3-cyclopropyl-4-[(pyrimidin-2-yl)amino]pyrrolidin-1-yl]-3-methanesulfonylpropan-1-one
4-{8-cyclopentyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-2-carboxylic acid
5-(2,3-dihydro-1-benzofuran-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-4H-1,2,4-triazol-4-amine
8-(5-chloropyridin-2-yl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-2-phenyl-7-[(2R)-pyrrolidine-2-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[2-(3-methoxyphenoxy)ethyl]-N-methyl-2-(2-oxoazonan-1-yl)acetamide
methyl (2S,4R)-1-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}-4-hydroxypyrrolidine-2-carboxylate
9-{[4-(2-aminoethyl)phenyl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
5-[2-(3-aminoazepan-1-yl)-2-oxoethyl]-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]pyrrolidine-1-carboxamide
N-(propan-2-yl)-1-(2-{4-[2-(trifluoromethoxy)benzenesulfonyl]piperazin-1-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
2-chloro-4-({ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}amino)benzamide
{4-[(4-chlorophenyl)methyl]-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-4-yl}methanol
3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidine
2-(2H-1,3-benzodioxol-5-yl)-N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)acetamide
3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]quinoline
1-(azepan-1-yl)-3-{3-[(4-methoxypiperidin-1-yl)methyl]phenoxy}propan-2-ol
[(2R)-1-{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}pyrrolidin-2-yl]methanol
5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-N-[(2R)-pyrrolidin-2-ylmethyl]pyridin-2-amine
(3R)-1-(2-ethoxybenzoyl)-3,4,4-trimethylpyrrolidin-3-ol
2-(adamantan-1-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
1-[4-({4-[3-(azocan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)-1,4-diazepan-1-yl]ethan-1-one
4-hydroxy-N-{1-oxaspiro[4.5]decan-3-yl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide
7-(cyclopropylmethyl)-2-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
1-[1-(2-carbamoylethyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
N-(2-ethyl-6-methylphenyl)-4-[(1-methylpiperidin-3-yl)methyl]piperazine-1-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methylbenzamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-[3-(pyridin-3-yl)phenyl]propanamide