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N-(2-fluorophenyl)-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-(hydroxymethyl)piperidin-3-ol
1-cycloheptyl-5-[4-(methoxymethyl)piperidine-1-carbonyl]piperidin-2-one
(1S,3R)-3-amino-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}cyclopentane-1-carboxamide
1-(4-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
ethyl 1-[(6-methoxy-2H-chromen-3-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-methoxy-3-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)pyrazine
ethyl 3-{[7-acetyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propanoate
5-{2-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-3-propylimidazolidine-2,4-dione
2-[3-(furan-2-yl)-1H-pyrazol-1-yl]-N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}acetamide
2-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)thiophen-3-amine
7-(1-benzothiophen-3-yl)-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-1-(2-methylphenyl)piperazin-2-one
N-[(1R,3R)-3-aminocyclopentyl]-4-methyl-2-(propan-2-yl)pyrimidine-5-carboxamide
2-[1-(3-benzyl-1H-1,2,4-triazol-5-yl)propyl]-2,3-dihydro-1H-isoindol-1-one
1-{1-[(4-acetamidophenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
N,N-dimethyl-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]aniline
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-methylpiperidin-2-one
ethyl 4-{4-[2-(4-fluorophenyl)ethyl]-3-oxo-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl}piperazine-1-carboxylate
4-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-3-(3,4,5-trimethoxyphenyl)-1H-pyrazole
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-4-(methylsulfanyl)benzamide
6-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 6-(4-methylpentanoyl)-2-[(2-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-methoxy-N-[2-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethyl]benzene-1-sulfonamide
2-{1-[5-(3-fluorophenoxymethyl)-1H-pyrazol-3-yl]-N-methylformamido}-N-methylacetamide
1-cyclopropyl-N-[2-(1H-imidazol-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
{4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
(1S,5R)-6-(cyclobutylmethyl)-3-(7-methyl-1-benzofuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3S,4R)-1-[(3,5-dichloropyridin-4-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
2-[(4-chlorophenyl)sulfanyl]-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-(pyrrolidin-1-yl)benzamide
1-{2-oxo-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
1-[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-2-(oxolan-2-yl)-1H-1,3-benzodiazole
N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-4-(pyridin-4-yl)pyrimidin-2-amine
6-(oxolan-2-yl)-2-(2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}phenyl)-3,4-dihydropyrimidin-4-one
3-[(2-methoxyethyl)sulfamoyl]-5-(2-methoxyphenyl)benzoic acid
(5S,9aS,9bS)-5-(2,1,3-benzothiadiazol-5-yl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
5-{[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-N-methylfuran-2-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
N-(3-phenyl-1,2,4-thiadiazol-5-yl)-4-(pyridin-3-yl)piperazine-1-carboxamide
1-(4-acetylpiperazin-1-yl)-3-(2-chlorophenyl)-3-(3-hydroxyphenyl)propan-1-one
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-(quinoxalin-2-yl)piperidin-4-ol
[7-fluoro-5-(5-fluoro-3,8-dimethylquinolin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
7-methyl-2-{2-[4-(methylsulfanyl)phenyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)(quinolin-8-ylmethyl)amine
2-[(4-chlorophenyl)methyl]-8-(6-ethyl-2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine