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2-{2-[(5-ethyl-1,3,4-oxadiazol-2-yl)amino]ethyl}-6-phenyl-2,3-dihydropyridazin-3-one
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
6-[(3,4-dimethoxypyridin-2-yl)methyl]-5,6-dihydro-1,6-naphthyridin-5-one
6-(methoxymethyl)-1-methyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{2-[(2S)-pyrrolidin-2-yl]ethyl}-5,6,7,8-tetrahydroquinoline-3-carboxamide
N-{1-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylpyridine-2-carboxamide
6-{[(3R,4S)-1-(cyclopropanesulfonyl)-4-propylpyrrolidin-3-yl]amino}pyrazine-2-carboxamide
1-(5-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophen-2-yl)-2-methylpropan-1-one
2-(1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperidin-2-yl)pyridine
1-(2-cyclohexylethyl)-3-({[(2,6-dimethylpyridin-4-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
methyl 2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-6-[3-(methylsulfanyl)propanoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-3,5-dimethoxybenzamide
6-oxo-N-(propan-2-yl)-N-[(2,4,5-trimethoxyphenyl)methyl]-1,6-dihydropyridine-3-carboxamide
1-[4-(piperidin-3-yl)benzoyl]azepane
5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidine
1-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-5,5-diphenylpiperidin-2-one
3,5-dimethyl-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)-1,2-oxazole-4-carboxamide
2-{2-[2-(1H-imidazol-4-ylmethyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
4-(2,3-dimethoxyphenyl)-5-(furan-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-[1-(4-chloro-1-ethyl-1H-pyrazol-5-yl)-N-ethylformamido]propanamide
(3R,4S)-4-(5-methylfuran-2-yl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}pyrrolidin-3-amine
2-{4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-1H-1,3-benzodiazole
9-(1-methyl-2-oxoimidazolidine-4-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-amine
1-(2-cyclopropylacetyl)-4-(2,3-dihydro-1H-inden-5-yloxy)piperidine-4-carboxylic acid
ethyl 2-[(butan-2-yl)(pyridin-3-ylmethyl)amino]acetate
N-benzyl-2-tert-butyl-N-[2-(dimethylamino)ethyl]-4-hydroxypyrimidine-5-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperazin-2-one
4-{[({2-[3-(4-methylpiperazin-1-yl)propoxy]phenyl}methyl)amino]methyl}-1,3-thiazol-2-amine
3-chloro-4-fluoro-N-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-benzothiophene-2-carboxamide
3-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}amine
N-cyclopentyl-2-(ethylamino)-N-(3-phenylprop-2-yn-1-yl)pyrimidine-5-carboxamide
N-(2-{7-[3-(1,3-benzothiazol-2-yl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
methyl 2-chloro-5-{[methyl({2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl})carbamoyl]amino}benzoate
2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)acetamide
N-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-6-oxa-9-azaspiro[4.5]decane-9-carboxamide
1,6-dimethyl-2-oxo-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
5-{[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-(methylsulfanyl)pyrimidine
3-ethyl-8-[(2-hydroxy-3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(2-methylphenyl)-1,4-diazepane
1-(2-methylbutyl)-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
5-cyclopropyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
3-[3-(cyclopropylmethyl)-5-[(2,3-difluorophenyl)methyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
1-(3-methoxyphenyl)-4-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]piperazin-2-one
2-({4-[4-(pyrimidin-4-yl)piperidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
2-(2-{2-[2-(2-methylphenyl)pyrimidin-5-yl]-1H-imidazol-1-yl}phenyl)ethan-1-ol