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(4aS,8aR)-1-(3-methoxypropyl)-6-(2-methylfuran-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
7-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,3-diazepane-2,4-dione
2-methoxy-3-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
4-({1-[2-(pyridin-2-yl)ethyl]piperidin-2-yl}methyl)morpholine
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2-(pyridin-2-ylsulfanyl)acetamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-5-ethylpyrimidin-2-amine
N-{2-cyclobutyl-7-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-1-methyl-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
N-(1-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methyl-3-(methylsulfanyl)propanamide
2-(cyclohex-1-en-1-yl)-1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-(cyclopropylmethyl)-3-hydroxy-3-[({[2-(trifluoromethyl)phenyl]methyl}amino)methyl]piperidin-2-one
5-chloro-6-(2,3-dimethoxyphenyl)pyridine-3-carboxylic acid
[1-(1,3-oxazole-4-carbonyl)piperidin-4-yl]diphenylmethanol
N-[(2-ethylpyrimidin-4-yl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}but-2-yn-1-one
2-benzyl-9-(1-methyl-2-oxoimidazolidine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
{[4-(butan-2-yloxy)-3-ethoxyphenyl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]azepan-4-amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4-fluorophenyl)methyl]piperidin-3-ol
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1-methylpiperidine-2-carboxamide
4-[(2E)-2-methylbut-2-en-1-yl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[(1S,5R)-6-[(5-cyano-1-ethyl-1H-pyrrol-3-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
(4aR,7aS)-1-acetyl-4-(3-chloro-5-methoxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]pyridine-2-carbonitrile
N-{2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-N-methylmethanesulfonamide
6,8-dichloro-3-(3-hydroxybutyl)-3,4-dihydroquinazolin-4-one
1-{[2-(benzyloxy)phenyl]methyl}piperidine-3-carbonitrile
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-[(3,4,5-trimethoxyphenyl)methyl]pyrrolidin-2-one
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2-(1H-pyrazol-1-yl)butanamide
5-(5-chloro-2-ethoxyphenyl)pyrazine-2-carboxylic acid
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
1-(oxan-4-yl)-4-(3-propyl-1H-pyrazole-5-carbonyl)piperazine
4-[3-(morpholine-4-carbonyl)piperidin-1-yl]-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-cyclobutanecarbonyl-N-{2-[(pyridin-3-yl)amino]ethyl}piperidine-4-carboxamide
4-(ethylamino)-N,5-dimethyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
(2R,3S,6R)-5-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
5-hydroxy-N-{1-[(4-methylphenyl)methyl]cyclopropyl}pyrazine-2-carboxamide
N-[2-fluoro-5-({[2-(3-phenylpyrrolidin-1-yl)ethyl]carbamoyl}amino)phenyl]acetamide
N-{6-methyl-3-oxo-1H,3H-furo[3,4-c]pyridin-4-yl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-hydroxyphenyl)ethan-1-one
5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[4-(3-methoxypropyl)piperidin-1-yl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-[(1-hydroxycyclohexyl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]urea
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(pyridine-4-carbonyl)pyrrolidin-3-yl]methanol
2-{2-[3-(benzyloxy)azetidin-1-yl]-2-oxoethyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
1-(2-{3-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}phenyl)ethan-1-one
N-(2,5-dimethylphenyl)-3-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}-3-oxopropanamide