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3-(3-methoxyphenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
ethyl 2-[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amino]-1,3-oxazole-4-carboxylate
3-{4-[2-(propan-2-yl)-1,3-benzoxazole-5-carbonyl]piperazin-1-yl}-1λ6-thiolane-1,1-dione
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
[(2-ethylpyrimidin-4-yl)methyl](methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
4-{4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperazin-1-yl}-2,6-dimethoxypyrimidine
3-{2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
1-{[1-tert-butyl-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-1H-1,2,3,4-tetrazole
(1S,5R)-3-(5-methoxyfuran-2-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(1,3-benzothiazol-2-yl)-2-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenol
6-amino-N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}pyridine-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(oxolane-2-carbonyl)piperidin-4-yl]propanamide
4-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine
1-(2-hydroxyethyl)-5-(3-methylfuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(3S,4S)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
3-ethyl-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[6,7-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-methyl-1,3-thiazole-4-carboxamide
2-(adamantan-1-yl)-4-hydroxy-N-(1-methylpiperidin-3-yl)pyrimidine-5-carboxamide
3-[3-(3,5-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-phenylpyrrolidine
(2S,4R)-1-cyclobutanecarbonyl-N-ethyl-4-(3-hydroxy-4-methylbenzamido)pyrrolidine-2-carboxamide
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]pyridin-2-amine
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
2-(piperidine-1-carbonyl)-6-[4-(1H-pyrazol-5-yl)phenyl]pyrazine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]thiolan-3-amine
1-{1'-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
3,5-dimethyl-N-[(3S,5S)-1-methyl-5-[(pyridin-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1,2-oxazole-4-carboxamide
5-({[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amino}methyl)-2-methoxyphenol
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
2-[(1S,5R)-3-(3-chlorobenzoyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
5-{4-[(2,5-dimethoxyphenyl)methyl]piperazine-1-carbonyl}-2-ethylpyrimidine
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3-{3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-2H-indazole
2-acetyl-8-[(3,5-dimethylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-N-(2,6-dimethylphenyl)benzamide
methyl({[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl})[(4-methylphenyl)methyl]amine
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-3-(benzyloxy)piperidine
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-3-(methanesulfonylmethyl)piperidine
1-cyclohexyl-3-(furan-2-yl)-5-[3-(1H-imidazol-1-yl)propyl]-1H-1,2,4-triazole
N-[(3S,4R)-1-(5-methyl-1,3-benzoxazol-2-yl)-4-propylpyrrolidin-3-yl]methanesulfonamide
4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]benzonitrile
3-(3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-2H-chromen-2-one
1-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridine-2-carbonyl]cyclopropane-1-carboxamide
2-amino-4-[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-(2H-1,3-benzodioxol-5-yl)-2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine-4-carboxamide
(1R,5R)-3-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-1-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-4-yl]piperidine-4-carboxamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
8-methoxy-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(morpholin-4-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}pyrimidine-5-carboxamide