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1-(2,2-dimethylpropyl)-4-({[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)pyrrolidin-2-one
3-[(1S,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propanamide
1-(6-methoxypyridin-3-yl)-3-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}urea
(3R,4R)-1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-[methyl(1,2-oxazol-3-ylmethyl)amino]-2-[2-(trifluoromethoxy)phenyl]acetic acid
8-(2-carboxybenzenesulfonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(4-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}phenyl)methanol
6-(2,3-dimethoxy-5-methylphenyl)pyrimidin-4-amine
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
3-[(3R,4S)-1-{imidazo[1,2-a]pyridine-3-carbonyl}-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
[(1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methyl]dimethylamine
1-(2-methylbutyl)-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
ethyl 5-(cyclohex-3-ene-1-carbonyl)-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-ethyl-N-(2-methylprop-2-en-1-yl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-(6-methoxyquinolin-8-yl)-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
4-[3-(4-cyclopentylpiperazine-1-carbonyl)phenyl]-2-methylbutan-2-ol
N-[2-(1H-imidazol-1-yl)ethyl]-7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{3-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propyl}-1H-indole
4-{[4-(3-chloro-1-benzothiophen-2-yl)-1H-1,2,3-triazol-1-yl]methyl}pyridine
6-tert-butyl-N-(furan-3-ylmethyl)-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(2,6-dimethylpyridin-3-yl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)pyrimidin-2-amine
N-[2-(4-fluorophenyl)ethyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(dimethylamino)-8-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
(3S,5S)-5-(cyclopropylcarbamoyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-3-carboxylic acid
N-methyl-5-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
8-(2,3-dimethoxybenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](ethyl)[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
3-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
2-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[1-(6-chloro-8-methylquinolin-4-yl)piperidin-4-yl]methyl}acetamide
N-(dimethyl-1,2-oxazol-4-yl)-4-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}benzamide
3-methyl-7-{2-[2-(trifluoromethyl)phenyl]acetyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-benzyl-3-butyl-1-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(diethylamino)-3-(2-methoxy-5-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}phenoxy)propan-2-ol
ethyl 1-(2,5-dimethylfuran-3-carbonyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
ethyl 1-[2-(2-methoxyphenoxy)acetyl]-4-(2-phenylethyl)piperidine-4-carboxylate
{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-[1-(2,6-dimethylphenoxy)propan-2-yl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(2R,3R)-3-amino-1'-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-tert-butyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1,3,4-oxadiazol-2-amine
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
5-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1H-indole
4-chloro-2-[(1E)-3-[4-(2,6-diaminopyrimidin-4-yl)piperazin-1-yl]-2-methylprop-1-en-1-yl]phenol
2-{2-[3-(3-methylphenoxy)azetidin-1-yl]-2-oxoethyl}-2-azaspiro[4.5]decan-3-one
6-[(3-methyl-1-benzofuran-2-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-[5-(1-phenylcyclopentanecarbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]-1H-pyrazole