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ethyl 2-{[2-(1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]amino}propanoate
2-(1-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}ethyl)phenol
(4aS,8aR)-1-[2-(5-methylfuran-2-yl)ethyl]-6-(6-methylpyridazin-3-yl)-decahydro-1,6-naphthyridin-2-one
4-(1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)morpholine
1-[2-(dimethylamino)ethyl]-5-oxo-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]pyrrolidine-3-carboxamide
2-(2-hydroxyethyl)-8-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2,2-dimethyloxan-4-yl)-1,3-oxazole-4-carboxamide
1-{5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-yl}-4-(oxan-4-yl)piperazine
[1-methyl-4-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperazin-2-yl]methanol
(1S,5R)-6-(1,3-thiazol-4-ylmethyl)-3-{thieno[3,2-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(1-methyl-1H-pyrrol-2-yl)-N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-2-oxoacetamide
(2-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)urea
2-benzyl-8-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
8-methoxy-N-{3-[(pyridin-3-yl)amino]propyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(3S,4S)-1-(5-methyl-1,2,4-oxadiazol-3-yl)-4-propylpyrrolidine-3-carboxylic acid
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-[3-(1H-pyrazol-1-yl)propyl]benzamide
1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
dimethyl({4-[(2E)-3-phenylprop-2-en-1-yl]-1,4-oxazepan-6-yl}methyl)amine
(2S)-1-acetyl-N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyrrolidine-2-carboxamide
1-(4-methylphenyl)-4-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)piperazin-2-one
1-[1'-(4-methylpyrimidine-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
4-chloro-1-methyl-3-{[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}-1H-indazole
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine-3-carboxylate
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,2-oxazole-5-carboxamide
(1R,5R)-6-[4-(difluoromethoxy)benzoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
7-methoxy-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-acetyl-N-(1H-1,3-benzodiazol-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)morpholine
4-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
N-(2-hydroxyethyl)-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
3-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-1-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}urea
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(1,2-oxazol-3-ylmethyl)-1H-pyrazole-3-carboxamide
4-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]morpholine
9-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3,9-diazaspiro[5.6]dodecane
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-[(dimethylcarbamoyl)amino]acetamide
4-[(2S,4R)-1-[(4-ethylphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
4-(2-methoxy-5-methylphenyl)-3-[2-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazole
N-benzyl-5-(4-methyl-1H-pyrazol-1-yl)furan-2-carboxamide
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-4-(1H-pyrazol-3-yl)benzamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-[(3-chlorophenyl)methyl]-N-(3-methoxypropyl)-1,3-benzoxazole-6-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)pyrazine-2-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-5-(1H-imidazol-1-ylmethyl)furan-2-carboxamide
1-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-N-methylpiperidine-2-carboxamide
methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-({4-[(6-methylpyridazin-3-yl)carbamoyl]phenyl}methyl)piperidine-3-carboxamide
N-cyclopentyl-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-cyclopropyl-N-(1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
N-(3,4-difluorophenyl)-1-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}piperidin-3-amine