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(5S)-5-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(pyridin-4-ylmethyl)amino)methyl]pyrrolidin-2-one
2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]pyrazine
(3S,4S)-4-[(dimethylamino)methyl]-1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-3-ol
2-methyl-4-[3-(4-phenyl-1,4-diazepane-1-carbonyl)phenyl]butan-2-ol
4-(2H-1,3-benzodioxol-5-ylmethyl)-3-oxo-N-(1-propyl-1H-1,2,4-triazol-3-yl)piperazine-1-carboxamide
3-[2-(4-fluorophenyl)ethyl]-1-(1H-pyrrole-2-carbonyl)piperidine
8-(4-aminopyrimidin-2-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-hydroxycyclohexyl)methyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(6-chloropyridin-3-yl)acetamide
3-{[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]amino}-N-(pyridin-3-yl)propanamide
6-(4-{2-[4-(propan-2-yl)morpholin-2-yl]acetyl}piperazin-1-yl)pyridine-3-carbonitrile
2-[2-(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
5-({[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]carbamoyl}amino)-2-fluoro-N-methylbenzamide
N-methyl-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2-{2-[1-(2,4-difluorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]ethyl}pyrazine
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(4-ethyl-5-methylthiophene-3-carbonyl)piperidine
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1H-pyrrole-2-carboxamide
2-(4-fluorophenyl)-1-[3-(2-methylphenoxy)azetidin-1-yl]ethan-1-one
2-(4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
2-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-6-methylimidazo[1,2-a]pyridine
2-(1H-imidazol-2-yl)-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]benzamide
1-[2-(4-chlorobenzenesulfonamido)ethyl]-3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)urea
2-[5-(1-methyl-4-phenylpiperidin-4-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
methyl 4-{[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl}benzoate
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(2-methylpentyl)piperidine
1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-ethyl-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
2-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane
{1-[2-(3-phenylpropyl)-1,3-benzoxazole-5-carbonyl]piperidin-3-yl}methanol
N-[2-(7-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-3-carboxamide
methyl 3-{2-[(benzylsulfamoyl)amino]ethoxy}benzoate
(3aR,6aR)-2-(oxan-4-yl)-5-(1,2-oxazole-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3R,4S)-1-(2-fluoro-6-methoxybenzoyl)-4-propylpyrrolidin-3-yl]acetamide
2-[(4-fluoro-2-methoxyphenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
7-cyclohexyl-2-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-[1-(3-phenyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]pyridine
1-[(2,2-dimethyloxan-4-yl)methyl]-3-(2-fluorophenoxy)azetidine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-methylpyridine-2-carboxamide
N-[(5-fluoro-2-oxo-2,3-dihydro-1H-indol-3-yl)methyl]-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
1-(4-tert-butylphenyl)-N-[(2-methyl-1H-imidazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-[4-(2-ethylbutyl)piperazin-1-yl]-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(azepane-1-carbonyl)-1-ethyl-N-[2-(1H-indol-3-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
8-benzyl-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(morpholin-4-yl)ethyl]-4-(4-{[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}piperidin-1-yl)benzamide
1-(2-{[6-(2-methoxyphenyl)pyridazin-3-yl]amino}ethyl)piperidin-4-ol
4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(methylsulfanyl)pyrimidine
N,1-dimethyl-6-oxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,6-dihydropyridazine-3-carboxamide
N-[1-(2,8-dimethylquinoline-4-carbonyl)piperidin-4-yl]pyridin-2-amine
4-[1-(2-chloro-6-fluorobenzoyl)azetidin-3-yl]pyridine
3-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methyl-1,2,4-oxadiazole-5-carboxamide
2-phenyl-5-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-pyrazol-3-one