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1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-3-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)urea
3-(1-methylpiperidin-3-yl)-1-(4-phenyl-1,4-diazepan-1-yl)propan-1-one
(2S)-2-{[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-2-phenylethan-1-ol
N-[2-(furan-2-yl)ethyl]-2-(2-oxopiperidin-1-yl)acetamide
1-(3-methylpyridin-2-yl)-4-[4-(piperidin-1-ylmethyl)benzoyl]piperazine
3-[2-(azocan-1-yl)-2-oxoethyl]-4-(cyclohexylmethyl)piperazin-2-one
1-(1'-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
(1S,4R)-2-[(4-methylnaphthalen-1-yl)methyl]-2-azabicyclo[2.2.1]heptan-3-one
N-methyl-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyrimidin-2-amine
2-amino-4-(3-methoxyphenyl)-6-[4-(morpholin-4-yl)phenyl]pyridine-3-carbonitrile
2-{9-[(4-fluorophenyl)carbamoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-{7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-[2-(2-methylphenyl)ethyl]piperidine
N-{1-[(4-methylphenyl)methyl]cyclopropyl}-2-(2-oxopyrrolidin-1-yl)propanamide
1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-4-(4-methyl-1H-pyrazol-3-yl)piperidine
6-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
3-[(1-cyclohexyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)methyl]-2,3-dihydro-1λ6-thiophene-1,1-dione
(2S)-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-acetamidopropanamide
1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(1H-pyrazol-1-yl)propan-1-one
2-ethyl-4-[(4-methyl-3-phenylpiperazin-1-yl)methyl]pyrimidine
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(pyridin-4-yl)quinoline-4-carboxamide
1-methyl-N-[2-methyl-1-(pyridin-2-yl)propyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-[1-(3-methylbut-2-en-1-yl)-4-(quinolin-6-ylmethyl)piperazin-2-yl]ethan-1-ol
4-(1H-imidazol-1-yl)-1-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperidine-4-carboxylic acid
2-{2-[1-(5-propyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
methyl 2-(4-{3-[(pyridin-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidin-1-yl)acetate
3-acetamido-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylthiophene-2-carboxamide
1-{2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
5-(4-phenylpiperidine-1-carbonyl)-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
1-(2-cycloheptylethyl)-3-(dimethyl-1H-1,2,4-triazol-3-yl)urea
1-(2-{3-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-3-methylimidazolidin-2-one
(2E)-N-{[3-methyl-7-(1,2,5-thiadiazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenylprop-2-enamide
methyl({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)(pyridin-2-ylmethyl)amine
5-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N-propylpyrimidin-2-amine
1-[3-(3-methoxypropyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
2-(4-fluorophenyl)-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-2-(morpholin-3-yl)acetamide
3-(3-methoxyphenyl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-pyrazole-4-carboxamide
8-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methoxy}quinoline-2-carboxamide
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-2-(1-methyl-1H-indol-3-yl)ethan-1-one
ethyl 1-[(2-methyl-1,3-thiazol-5-yl)methyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
2-(3-methoxypropyl)-9-(3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(furan-2-ylmethyl)-4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
N-[5-({4-[(3-chlorophenyl)methyl]-5-oxo-1,4-diazepan-1-yl}methyl)thiophen-2-yl]acetamide
N-cyclopentyl-1-[1-(2,2-dimethylpropyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
1-(4-{[(2-methoxyethyl)[(4-methylphenyl)methyl]amino]methyl}phenyl)ethan-1-one
4-methoxy-N-{[1-(pyridine-2-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
4-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one