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methyl 6-({[(5-chloro-2-methoxyphenyl)methyl](ethyl)amino}methyl)pyridine-2-carboxylate
1-(piperidin-1-yl)-3-{4-[({2-[4-(trifluoromethyl)phenyl]ethyl}amino)methyl]phenoxy}propan-2-ol
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
1-methyl-3-propyl-N-[3-(pyridin-2-yl)propyl]-1H-pyrazole-5-carboxamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2-(dimethyl-1,3-thiazol-5-yl)acetamide
4-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}morpholine
7-methyl-3-{[methyl(pyridin-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
N-(2-ethyl-1,3-dihydroxypropan-2-yl)-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(2-{[2-amino-6-(propan-2-yl)pyrimidin-4-yl](methyl)amino}ethyl)cyclopentan-1-ol
3-[2-(2-methylpropanesulfonyl)ethyl]-1-[3-(methylsulfanyl)phenyl]urea
(4aR,8aS)-6-(3-fluorobenzoyl)-1-[(2-methoxyphenyl)methyl]-decahydro-1,6-naphthyridine
N-butyl-1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]propanamide
N-cyclooctyl-1-(2-methoxyethyl)-4-oxo-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
5-ethyl-4-[4-(2,2,2-trifluoroethyl)piperazin-1-yl]pyrimidin-2-amine
N-ethyl-3-{imidazo[1,2-a]pyridin-2-yl}-N-(2-methylprop-2-en-1-yl)propanamide
4-(furan-3-ylmethyl)-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperazin-2-one
[(1-{1-[1-(2-fluorophenyl)piperidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl](methyl)amine
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]propanamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
1-(2-aminopyrimidin-4-yl)-3-[(2,4-difluorophenyl)methyl]piperidine-3-carboxylic acid
2,6-diamino-4-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
5,6-dimethyl-3-[4-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-benzyl-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}pyrrolidin-3-amine
6-ethyl-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-2-methylquinoline-4-carboxamide
[3-(1H-imidazol-1-yl)propyl]({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})(pyridin-4-ylmethyl)amine
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
methyl 3-cyclobutaneamido-5-{[(2-fluorophenyl)methyl]amino}-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[(1S,2R)-1-hydroxy-2-{4-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}propyl]phenol
1-{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}piperidin-3-ol
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-methyl-2-phenylpropan-1-one
2-methoxy-N-{[5-(quinolin-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
methyl 4-{[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[1-(cyclohexylmethyl)-5-[5-(pyrrolidin-1-ylmethyl)furan-2-yl]-1H-1,2,4-triazol-3-yl]acetamide
1-[(2-methoxypyridin-3-yl)methyl]-3-methyl-1,2-dihydroquinoxalin-2-one
N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-2-(4-phenylphenyl)acetamide
3-(2H-1,3-benzodioxol-5-yl)-5-(2,3-dihydro-1H-inden-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-acetyl-8-[2-(4-chlorophenoxy)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{[1-(1H-indol-2-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
9-(2,6-dimethylpyrimidine-4-carbonyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(2R)-4-[5-(2-ethylphenyl)-4-phenyl-1H-imidazol-1-yl]-2-methylbutan-1-ol
7-[4-(1-ethoxyethyl)phenyl]-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
N-(3-phenylphenyl)-4-(pyrrolidine-1-carbonyl)piperidine-1-carboxamide
2-(4-hydroxy-3-methoxyphenyl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(1,3-benzothiazol-2-ylmethyl)-1-ethyl-N-methyl-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(1,3-dihydro-2-benzofuran-5-yl)-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
(4aR,7aS)-1-(2-methoxyacetyl)-4-(1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(3,4-dimethylphenoxy)propyl]-N-methyl-3-(1,2-oxazolidin-2-yl)propanamide
(2R,3R,6R)-3-(4-methylphenyl)-5-(6-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane