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6-methyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
N-(2-hydroxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-6-carboxamide
4-[(5-acetylthiophen-3-yl)methyl]-N,N-dimethylpiperazine-1-sulfonamide
1-methyl-N-[(3-methylphenyl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
4,6-dimethyl-2-[4-(pyrrolidine-1-carbonyl)phenyl]pyridine-3-carboxamide
4-[4-(diethylamino)-2-hydroxyphenyl]-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]benzamide
1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyloxane-4-carboxamide
N-[4-(pyridin-2-yl)butyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-({1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}methyl)-4-phenylbenzamide
5-[3-(4-fluorophenyl)-1H-pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N3-(2H-1,3-benzodioxol-5-ylmethyl)-N5-butyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-4-(trifluoromethyl)benzamide
N-methyl-2-{4-[(2-methylphenyl)methyl]-2,5-dioxo-4-(piperidin-4-yl)imidazolidin-1-yl}acetamide
7-[(2S)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
3-(3-chlorophenyl)-1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)pyrrolidine
3-{[(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)amino]methyl}pyrrolidin-3-ol
2-(benzylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-(pyridin-2-yl)-1-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
6-chloro-3-fluoro-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]imidazo[1,2-a]pyridine-2-carboxamide
4-({4-[1-(dimethylamino)ethyl]piperidin-1-yl}methyl)-1-ethyl-1H-pyrrole-2-carbonitrile
4,6-dimethyl-2-oxo-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-(2,5-dimethyl-3-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)acetamide
ethyl 4-(4-{2-[(1-hydroxycyclohexyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperazin-1-yl)piperidine-1-carboxylate
1-[(4aR,8aR)-4a-hydroxy-7-(4-propylbenzoyl)-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
(1R,6S)-9-methyl-3-(2-propoxybenzoyl)-3,9-diazabicyclo[4.2.1]nonane
2-(4-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-2-oxopiperazin-1-yl)benzonitrile
N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-2-(1-propylpiperidin-4-yl)acetamide
8-methoxy-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-methyl-4-{3-[2-(pyridin-4-yl)-1H-imidazol-1-yl]phenyl}pyrimidine
N-{2-methyl-4-[3-(1H-pyrazol-3-yl)phenyl]phenyl}pyridine-3-carboxamide
(3S,4R)-3-methoxy-1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-4-amine
4-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-3-yl]-2-methyl-5-(3-methylphenyl)pyrimidine
4-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1H-imidazol-2-yl}-2-(propan-2-yl)pyrimidine
N-(3-phenylpropyl)-N-(propan-2-yl)quinoxaline-5-carboxamide
1-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)urea
5,6-dimethyl-2-(2-{[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}ethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
(3R,4R)-4-ethyl-1-(5-methyl-2-phenylfuran-3-carbonyl)piperidine-3,4-diol
N-[2-chloro-5-(diethylcarbamoyl)phenyl]-5-methylpyridine-3-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]propanamide
2-(cyclopropylmethyl)-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3aS,6aS)-2-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(1-benzylpyrrolidin-3-yl)-3-[1-(3-fluorobenzoyl)piperidin-4-yl]propanamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[2-phenyl-2-(piperidin-1-yl)ethyl]acetamide
2,4,5-trimethyl-6-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyrimidine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-1-(oxan-4-yl)piperidine-4-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-N-propyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide