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1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-4-(azepan-1-yl)butane-1,4-dione
8-cyclopropanecarbonyl-2-(4-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[3-(ethoxymethyl)-5-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-3-phenyl-1H-pyrazole-4-carboxamide
6-[(diethylamino)methyl]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]amine
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepan-5-one
(4aS,7aR)-1-(3-methyl-1H-pyrazole-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(1-methyl-1H-indole-6-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[(1R,5S,6S)-3-[2-(benzyloxy)ethyl]-3-azabicyclo[3.1.0]hexane-6-carbonyl]piperidin-4-ol
N,4-dimethyl-6-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
1-{4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
4-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]pyrimidin-2-amine
8-(3-fluoro-4-methoxybenzoyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-{[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}-1,4-oxazepan-6-ol
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
2-(4-chlorophenyl)-4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)morpholine
4-(2-amino-6-methylpyrimidin-4-yl)-N-benzylpiperazine-1-sulfonamide
6-fluoro-N-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(oxan-2-ylmethyl)quinoline-4-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid
1-(5-{1H-pyrazolo[3,4-b]pyridin-1-yl}-1H-1,3-benzodiazol-2-yl)ethan-1-ol
4-(3-methoxyphenyl)-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]benzamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-cyclohexyl-N-(prop-2-yn-1-yl)-1,2-oxazole-3-carboxamide
2-{3-[1-(5-fluoropentyl)-1H-pyrazol-3-yl]phenyl}pyrazine
N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
2-{[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
N-benzyl-N-(2-hydroxyethyl)-2-(1H-pyrazol-1-yl)butanamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
N-({3-methyl-7-[4-(1H-pyrazol-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(phenylsulfanyl)acetamide
2-hydroxy-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-cyclohexyl-8-fluoro-N-(pyridin-4-ylmethyl)quinoline-2-carboxamide
4-phenyl-2-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,3-thiazole
5-chloro-3-[4-(1-hydroxy-3-methylbutyl)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-(2-hydroxyethyl)-8-[2-(4-hydroxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(pyridin-3-yl)propanamide
3-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-benzyl-4-({4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)piperazine
2-[(3R,4S)-3-[(6-cyclopropylpyrimidin-4-yl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]propane-1,3-diol
2-(4-chlorophenyl)-2-hydroxy-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]acetamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]ethan-1-one
(2S)-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}-2-(pyrrolidin-1-ylmethyl)pyrrolidine
8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
1-(4-cyclopentylpiperazin-1-yl)-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
N-(furan-2-ylmethyl)-1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidine-4-carboxamide
2-{2-[5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-2-oxopiperidin-1-yl]ethyl}-6-methyl-3,4-dihydropyrimidin-4-one
N-[2-(2-ethoxyphenoxy)ethyl]-N-methyl-5-(oxolan-2-yl)thiophene-2-carboxamide
N-[1-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)piperidin-4-yl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide