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(3S,7S)-5-(2-ethylpyrimidine-5-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
5,7-dimethyl-N-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)propyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-(2-phenylpropyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
2-{2-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
(3S,4S)-4-[4-(pyridin-2-yl)piperazin-1-yl]-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]pyrrolidin-3-ol
4-({8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1H-pyrazole-3-carboxylic acid
3-(1-{1-[4-(dimethylamino)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(3-fluorophenyl)urea
2-methyl-3-(1,4-oxazepane-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
N-(cyclohexylmethyl)-3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carboxamide
8-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-(2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}pyrimidin-4-yl)piperidin-4-ol
1-{2-[1-(3-chloro-4-methoxybenzoyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
4-(5-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
ethyl 4-({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)piperidine-1-carboxylate
7-fluoro-4-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[2-(6-methylpyridin-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(quinazolin-4-yl)amino]pentanamide
methyl 3-(furan-2-amido)-5-{[(2-methoxyphenyl)formamido]methyl}benzoate
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pyrimidine-4-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(methoxymethyl)-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
1-(2-methyl-1-benzofuran-7-yl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-methylpropyl)urea
2-(2-amino-4-methyl-1,3-thiazol-5-yl)-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}acetamide
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorothiophene-2-carboxamide
2-[4-({[1-(2-methoxyphenyl)ethyl](methyl)amino}methyl)phenyl]-5,6-dimethyl-3,4-dihydropyrimidin-4-one
5-ethyl-N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-benzyl-9-ethyl-2,9-diazaspiro[5.5]undecan-3-one
2-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridin-3-ol
[5-({cyclopropyl[(3-methylthiophen-2-yl)methyl]amino}methyl)furan-2-yl]methanol
3-(3-{furo[3,2-c]pyridin-4-yl}phenyl)-1H-pyrazole
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-2-phenylethan-1-one
N-(2-hydroxyethyl)-5-[1-(piperidin-1-yl)ethyl]-N-(1,3-thiazol-2-ylmethyl)furan-2-carboxamide
4-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
(2R,6R)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-[2-(4-methylphenoxy)propan-2-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-(2-methyl-1H-pyrrole-3-carbonyl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
3-methyl-4-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-ethyl-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)morpholine-2-carboxamide
2-[1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1H-pyrazol-4-yl]ethan-1-ol
3-ethoxy-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methyl-4-(prop-2-en-1-yloxy)benzamide
3-(3-fluoro-4-phenylbenzoyl)-1-(1,2-oxazol-3-ylmethyl)piperidine
(3R,5R)-1-(naphthalen-2-ylmethyl)-3-(pyrrolidin-1-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-6-methylpyrimidin-2-amine
(1R,2R,4R)-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
(1S,5R)-3-(oxan-4-yl)-6-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
1-({1-[6-(pyridin-4-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
[3-ethyl-1-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)piperidin-3-yl]methanol
1-{3-[3-(quinolin-2-yl)phenyl]-1H-pyrazol-1-yl}butan-2-ol