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3-(piperidin-3-yl)-N-{[1-(pyrrolidin-1-yl)cyclohexyl]methyl}benzamide
1-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
2-(2-methoxy-4-methylphenoxymethyl)-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}bis(prop-2-en-1-yl)amine
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-8-methoxy-1,2,3,4-tetrahydroquinolin-2-one
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1H-indole-5-carboxamide
8-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(3-{2-[(4-fluoropiperidin-1-yl)methyl]-4-methoxyphenoxy}-2-hydroxypropyl)piperidin-4-ol
N'-(3,5-dimethylphenyl)-N-methyl-N-[2-(morpholin-4-yl)propyl]propanediamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(2-oxopiperidin-1-yl)propanamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-(furan-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methoxy-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenol
5-oxo-1-(pyridin-4-ylmethyl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-3-carboxamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-tert-butyl-7-[(2H-1,2,3,4-tetrazol-5-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-(3-{[3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propyl)pyrrolidin-2-one
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(3-hydroxyphenyl)methyl]piperidin-3-yl]propanoate
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carbonitrile
N-(4-fluorophenyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-3-amine
5-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-2-methylpyrimidine
3-(3-hydroxy-3-methylbutyl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}benzamide
(4aS,7aR)-1-[2-(dimethylamino)benzoyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2-methylpyrimidin-4-yl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{[(propan-2-yl)(quinolin-2-ylmethyl)amino]methyl}pyrrolidin-2-one
6-(1-methyl-1H-imidazol-2-yl)-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)pyridazin-3-amine
6-(benzyloxy)-1-cyclohexyl-4-(1-ethyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-2-one
N-[2-(1H-imidazol-4-yl)ethyl]-6-(2-methoxyphenyl)pyridazin-3-amine
4-methoxy-6-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]pyrimidin-2-amine
1-(carbamoylmethyl)-N-[2-(4-fluorobenzenesulfonyl)ethyl]piperidine-3-carboxamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N,N-bis(1,3-oxazol-4-ylmethyl)acetamide
1-[4-(furan-2-yl)pyrimidin-2-yl]-N-[3-(morpholin-4-yl)propyl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-(1H-imidazol-2-ylmethyl)-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-{4-[1-(dimethylamino)ethyl]phenyl}-5-(morpholine-4-sulfonyl)benzoic acid
1'-(3-ethyl-1H-pyrazole-5-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[4-(methylsulfanyl)phenyl]ethan-1-one
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[2-(1H-pyrazol-1-yl)phenyl]piperazine-1-carboxamide
6-{[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
4-(2-methyl-1H-imidazol-1-yl)-1-(thiophen-2-ylmethyl)piperidine-4-carboxylic acid
1-(4-{[bis(prop-2-en-1-yl)amino]methyl}-2-methoxyphenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[3-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-oxopropyl]-4-methylbenzamide
3-[(3-chlorophenyl)methyl]-5-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-1-ethyl-1H-1,2,4-triazole
N-[2-(hydroxymethyl)phenyl]-4-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)benzamide
N-cyclopropyl-N-[(3-methylthiophen-2-yl)methyl]-2-(pyridin-3-yl)acetamide
(3aS,6aS)-2-methanesulfonyl-5-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aR,7aS)-1-(2-methylpropyl)-4-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[(2-fluorophenyl)methyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxy-2,2-dimethylpropyl)acetamide
3-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1-(2,6-dimethylpyridin-3-yl)urea
(1R,7S)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-oxo-3-(pentan-3-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide