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6-oxo-4-(1-phenyl-1H-pyrazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
(2S,3R)-3-hydroxy-2-[(2-{[4-(propan-2-yl)phenyl]carbamoyl}ethyl)amino]butanamide
8-methoxy-4-methyl-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
3-phenyl-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-{[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl}propanamide
1-[2-(2-methoxyethoxy)phenyl]-3-[2-(5-methylfuran-2-yl)ethyl]urea
1-[2-methoxy-4-({[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-[(1R,3R)-3-aminocyclopentyl]-2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
(3S)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperidine-3-carboxylic acid
2-(3-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}phenoxy)ethan-1-ol
(3R,9aR)-3-methyl-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methyl-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-2-(thiophen-2-ylformamido)propanamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]benzamide
methyl (2R,4S)-4-hydroxy-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidine-2-carboxylate
N-cyclohexyl-3-{[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]methyl}-N-methylpyridin-2-amine
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-ethylpyrrolidine-3-carboxamide
8-(4-chloro-2-methoxybenzoyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(pyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
7-[(2,3-difluorophenyl)methyl]-2-[(4-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
1-[(2,5-dimethoxyphenyl)methyl]-4-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazine
N-(1-methylpiperidin-4-yl)-2-(morpholin-2-yl)-N-(2-phenylethyl)acetamide
2-(3-chloro-2,6-difluorophenyl)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
3-(1,4-dioxan-2-ylmethyl)-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,4-dimethyl-1,2,5-oxadiazole-3-carboxamide
2-{5-[(1R,3S)-3-aminocyclohexyl]-3-(4-tert-butylphenoxymethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-(4,6-dimethoxypyrimidin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-amino-4-{[2-methyl-1-(pyridin-3-yl)propyl]amino}quinazoline-6-carboxylic acid
2-(naphthalen-1-yl)-1-{4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
2-(azepan-1-yl)-1-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}ethan-1-one
(1S,5R)-6-(1H-indole-2-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-benzyl-6-(4-methyl-1,4-diazepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(1S,5R)-N-benzyl-N,6-dimethyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-{5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}thiomorpholine
4-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-1-methyl-2-phenylpiperazine
1-ethyl-3-methyl-4-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}sulfonyl)-1H-pyrazole
(1S,5R)-3-{3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanoyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(3-fluorophenyl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}propanamide
3-[1-butyl-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]piperidine-1-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-1-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]propan-1-one
N-(3-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}phenyl)acetamide
(2S,4R)-4-[(2,3-dihydro-1H-inden-2-yl)amino]-N-[2-(2-fluorophenyl)ethyl]-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-{5-cyclopropyl-4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(2,5-dimethoxyphenyl)pyrimidine
4-[(1H-imidazol-2-ylmethyl)sulfamoyl]-N-[(3S)-pyrrolidin-3-yl]benzamide
9-(5-chloropyridin-2-yl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
2,4-dimethyl-6-[3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carbonitrile
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
2-(adamantan-1-yl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}acetamide
{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
4-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}-6-(pyrrolidin-1-yl)pyrimidin-2-amine