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N-[1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-phenoxypropanamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(3-phenylpropyl)-1,4-diazepane
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]propanamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-tert-butyl-4-hydroxypyrimidine-5-carboxamide
1-ethyl-4-{[methyl({[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
(2,1,3-benzoxadiazol-5-ylmethyl)[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
1,5-dimethyl-4-({4-[2-(phenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
3-{[(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
N-[2-(2-hydroxy-2-methylpropanamido)-4-methylphenyl]-2-methylbenzamide
7-fluoro-2-methyl-4-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]quinoline
N-(oxolan-2-ylmethyl)-N-propyl-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-(3-methyl-1,2,4-oxadiazol-5-yl)-1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidine
(4aR,6R,8aS)-8a-(methoxymethyl)-2-(2-methylpyrimidine-5-carbonyl)-6-(morpholin-4-yl)-decahydroisoquinoline
4-benzyl-3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-fluoro-3-(trifluoromethyl)phenyl]-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
1-[(4-chlorophenyl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-methyl-5-(morpholin-4-ylmethyl)-N-(2-phenylethyl)-1,2-oxazole-3-carboxamide
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-methoxyethan-1-one
(3aR,6aR)-2-methanesulfonyl-5-(3-methylthiophene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-hydroxy-5-[2-(morpholin-4-ylmethyl)phenyl]benzoic acid
(4aS,8aR)-1-(4-hydroxybutyl)-6-[(2E)-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
2-{1-[(2-ethoxypyridin-3-yl)methyl]-1H-imidazol-2-yl}-1-methyl-1H-1,3-benzodiazole
1-[2-methoxy-5-(thiomorpholin-4-ylmethyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
N-[(3S,4R)-1-(1,3-benzothiazol-2-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
2-(2-chloro-4-fluorophenyl)-5,6-dimethylpyridine-3-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-N-{[(propan-2-yl)carbamoyl]methyl}acetamide
1-cyclobutanecarbonyl-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-[2-(2,5-dimethylphenoxy)ethyl]piperidin-3-amine
1-{4-[({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}amino)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-ethyl-9-[2-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aR,7aS)-1-cyclobutanecarbonyl-4-(3-ethyl-1,2-oxazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{2-oxa-7-azaspiro[4.5]decan-7-yl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
{[2-(azocan-1-yl)pyridin-3-yl]methyl}[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amine
7-cyclohexyl-2-(6-methoxyhexanoyl)-2,7-diazaspiro[4.5]decan-6-one
2-(2,5-difluorophenyl)-1-{4-[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
4-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}-N-methylbenzene-1-sulfonamide
(3S)-1-[1-methyl-5-(3-phenoxyazetidine-1-carbonyl)-1H-1,3-benzodiazol-2-yl]pyrrolidin-3-ol
N-methyl-N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}naphthalene-2-sulfonamide
2-(ethylsulfanyl)-5-{[4-(4-fluorophenoxy)piperidin-1-yl]methyl}pyrimidine
(3aS,6aS)-2-(2-chloro-4-fluorobenzoyl)-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2-methyl-1H-1,3-benzodiazol-5-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
2-(4-chloro-1H-pyrazol-1-yl)-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)acetamide
N-methyl-N-[2-(4-methylphenoxy)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide