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3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenylurea
3-{[(2H-1,3-benzodioxol-4-ylmethyl)amino]methyl}-N,N-diethylpyridin-2-amine
2-(ethylamino)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]pyrimidine-5-carboxamide
2-(2-hydroxyethyl)-8-[4-(1H-pyrazol-4-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
3-[(cyclopentylmethyl)sulfamoyl]-N-(1,4-dioxan-2-ylmethyl)benzamide
4-(4-fluorophenoxy)-1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
7-(3,6-dimethylpyrazin-2-yl)-4-(piperidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2,3-dihydro-1H-indol-1-yl)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-oxoacetamide
1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-3-methylpiperazine
4-[4-(1H-pyrazol-5-yl)phenyl]pyridin-2-amine
ethyl 3-[(4-{2-[benzyl(methyl)carbamoyl]ethyl}piperidine-1-carbonyl)amino]propanoate
(2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
(4aS,8aR)-1-[2-(5-methylfuran-2-yl)ethyl]-6-(3-methylpyrazin-2-yl)-decahydro-1,6-naphthyridin-2-one
N-[3-(1H-imidazol-1-yl)propyl]-2-(methylamino)pyridine-4-carboxamide
1-(2-methoxyethyl)-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]piperidine
(2S)-2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-4-(methylsulfanyl)butan-1-ol
N-[2-(1H-imidazol-4-yl)ethyl]-2,2-dimethyloxane-4-carboxamide
N-cyclopropyl-4-methoxy-3-[(1-methylpiperidin-4-yl)oxy]benzamide
3-cyano-N-[(2-ethoxyphenyl)methyl]-N-ethylbenzamide
5-acetyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}thiophene-3-carboxamide
2-methoxy-1-{1'-[(3-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
2-{2-[(2,4-dimethyl-1,4-diazepan-1-yl)methyl]-4-(pyridin-2-yl)phenoxy}acetic acid
3-{[benzyl(methyl)amino]methyl}-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
3-[2-(azonan-1-yl)-2-oxoethyl]-4-(propan-2-yl)piperazin-2-one
5-cyclobutyl-N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-1,3,4-thiadiazol-2-amine
4-(5,6-dimethylpyrimidin-4-yl)-2-(2-methoxyethyl)morpholine
1-benzyl-8-[(3-hydroxyphenyl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(azepan-1-yl)-2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]ethane-1,2-dione
3-methyl-7-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-(carbamoylmethyl)-N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]piperidine-4-carboxamide
2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl](methyl)amino}ethan-1-ol
{4-[2-(methoxymethyl)-1,3-benzoxazol-5-yl]phenyl}methanol
(1R,5R)-3-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-(1-methoxybutan-2-yl)-1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(2-methoxyethyl)-1-(1H-1,2,3-triazole-5-carbonyl)piperidine-3-carboxylic acid
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]furan-2-carboxamide
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
8-(5-methylpyrazine-2-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
4-(azepan-1-yl)-4-oxo-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}butanamide
N-ethyl-3-[2-(3-fluorophenyl)ethyl]piperidine-1-carboxamide
6-methyl-3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]pyrazolo[1,5-a]pyrimidine
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-fluorophenyl)urea
1-[2-benzyl-4-(3-methoxyphenyl)-5-oxopiperazin-1-yl]propane-1,2-dione
2-fluoro-N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
ethyl 4-(oxan-2-ylmethyl)piperidine-4-carboxylate
N-(2,3-difluorophenyl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-N,N,5,6-tetramethylpyrimidin-2-amine