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2-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1,2-oxazolidin-4-ol
1-(4-fluorophenyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]-1,4-diazepane
(1S,5R)-6-benzyl-3-[(2-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(2,6-difluorophenyl)methyl]-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
4-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}oxane-4-carbonitrile
2-(4-methyl-1H-imidazol-5-yl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-imidazole
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-(oxolane-2-carbonyl)piperazine
1-[9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(2-methoxyphenyl)propan-1-one
N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)pent-4-enamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)benzamide
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(2-methylphenoxymethyl)piperidine
1-methyl-4-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(1-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)thiomorpholine
N3-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[2-(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
3-[(3R,4S)-1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
4-{[3-(azocan-1-yl)propanamido]methyl}benzoic acid
3-{5-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-(4-acetylphenyl)-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-6-methylphenol
(4aR,7aS)-1-methyl-4-[2-(1-methyl-1H-indol-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2,3-dimethyl-6-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-methyl-6-oxo-N-(propan-2-yl)-1,6-dihydropyridine-3-carboxamide
5-(2-chlorophenyl)-N-ethyl-2-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]furan-3-carboxamide
2-[4-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)piperazin-1-yl]pyrimidine
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(4-methyl-1H-imidazole-2-carbonyl)piperidine
2-{[6-(6-fluoroquinolin-8-yl)pyrazin-2-yl]sulfanyl}acetic acid
N-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]pyridin-2-amine
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-[(1-ethylpiperidin-4-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
9-(2-methoxyethyl)-1-methyl-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N'-(3-chloro-4-fluorophenyl)-N-[1-(furan-2-yl)ethyl]-N-methylpropanediamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-5-methyl-1,2-oxazole-4-carboxamide
8-(1-benzyl-1H-pyrazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2,6-diamino-4-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
methyl 5-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-(piperidine-1-carbonyl)pyrazin-2-amine
6-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-5-chloropyridine-3-carboxylic acid
3-({1-[2-(propan-2-ylsulfanyl)acetyl]pyrrolidin-3-yl}methyl)benzoic acid
2-[2-(cyclohex-1-en-1-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(2-{1-[2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N1-{2-methylthieno[2,3-d]pyrimidin-4-yl}ethane-1,2-diamine
N-{[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
2-methyl-4-(4-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}phenyl)but-3-yn-2-ol
2-(methoxymethyl)-5-{1-[1-(pyridin-4-yl)propan-2-yl]-1H-1,2,3-triazol-4-yl}pyrimidine
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-[1-(pyrazin-2-yl)propan-2-yl]urea