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(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-N-(2-chlorophenyl)-3-hydroxypiperidine-1-carboxamide
6-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]quinoline
1-cyclopentyl-N-methyl-N-(quinoxalin-2-ylmethyl)piperidine-3-carboxamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-(2,3-dihydro-1H-inden-2-yl)propanamide
[2-(morpholin-4-yl)ethyl]({[6-(thiophen-3-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
1-methyl-6-propyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
[1-(1-methylpyrrolidine-3-carbonyl)piperidin-4-yl]diphenylmethanol
ethyl 2-{1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-amido]cyclohexyl}acetate
4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-1-(cyclopropylmethyl)-2-(propan-2-yl)-1,4-diazepane
(4aR,8aR)-2-cyclobutanecarbonyl-7-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-decahydro-2,7-naphthyridin-4a-ol
5-cyclopropanecarbonyl-1'-(pyridin-4-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
(1R,5R)-N,N-dimethyl-6-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(2-methoxyethyl)-1-[1-(9H-purin-6-yl)piperidin-4-yl]piperidine-3-carboxamide
(3aS,6aR)-5-(4-hydroxybenzoyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
{1-[1-(2-methoxyethyl)piperidine-4-carbonyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
N-[(1-benzylpiperidin-4-yl)methyl]-5-chloro-N-methylpyridine-3-carboxamide
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(4-fluorophenyl)piperidin-4-ol
3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]-1-(thiophene-2-carbonyl)piperidine
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1-(carbamoylmethyl)piperidine-4-carboxamide
1-[2-(3,5-dichlorophenyl)-4-hydroxypyrimidine-5-carbonyl]piperidine-3-carboxamide
3-[(cycloheptylamino)methyl]-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
1-(2,3-difluorobenzoyl)-2-(4-fluorophenyl)piperidine
2-(1-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-3-yl)benzoic acid
N-methyl-N-{2-[4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}methanesulfonamide
N-[(2S,4R,6R)-2-[(benzyloxy)methyl]-6-(4-fluoro-3-methoxyphenyl)oxan-4-yl]acetamide
N-(2-methoxyethyl)-2,6-dimethyl-N-(1-methylpiperidin-4-yl)quinoline-3-carboxamide
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl){[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}amine
7-methyl-2-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-[(3-fluorophenyl)methyl]-N-[2-(naphthalen-1-yl)propan-2-yl]-6-oxopiperidine-3-carboxamide
4-(propan-2-yl)-N-[2-(pyridin-3-yloxy)propyl]pyrimidin-2-amine
1-[3-(aminomethyl)pyrrolidin-1-yl]-3-[5-(4-chlorophenyl)-1H-pyrrol-2-yl]propan-1-one
N-[(2-methoxyphenyl)methyl]-3-methyl-N-(pyridin-4-ylmethyl)-1,2-oxazole-5-carboxamide
5-[4-hydroxy-1-(thiophen-2-ylmethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
4-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-N-(1-methyl-1H-pyrazol-4-yl)benzamide
3-(1,4-diazepane-1-carbonyl)-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzene-1-sulfonamide
N3-cycloheptyl-1-cyclopropyl-4-oxo-N5-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-(4-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}phenyl)acetamide
5-[2-(4-methylpiperidin-1-yl)propanoyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-[3-(2-fluoro-6-methoxyphenyl)phenyl]-4H-1,2,4-triazole
N-{[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}-N-cyclopropyl-4-(morpholin-4-yl)benzamide
4-acetyl-5-benzyl-1-(3-methoxyphenyl)piperazin-2-one
4-{[1-(1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
1-[2-({2-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]imidazolidin-2-one
2-[3-(2-chlorophenyl)pyrrolidin-1-yl]-5-cyclopropyl-1,3,4-oxadiazole
N-({7-[2-(1H-indol-3-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
(4aS,7aR)-1-(3-methylbutyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-[(3S,4R)-1-benzyl-4-(4-methylpiperazin-1-yl)piperidin-3-yl]-N-[2-(1H-indol-3-yl)ethyl]propanamide
3-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenol