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1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-methyl-3-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)imidazolidin-2-one
4-ethyl-3-(1-hexanoylpiperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2,5-dioxoimidazolidin-4-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}acetamide
N-[2-(4-methoxyphenyl)ethyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1'-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)spiro[indene-1,4'-piperidine]
N,1-dimethyl-6-propyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(dimethylamino)-2-[(3-fluorophenyl)methyl]-2,3-dihydropyridazin-3-one
N-methyl-5-phenyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1,2-oxazole-3-carboxamide
(3aR,6aR)-2-methanesulfonyl-5-(3-methylbutyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2'-amino-4'-(1-methyl-1H-pyrazol-4-yl)-7',8'-dihydro-5'H-spiro[piperidine-4,6'-quinoline]-3'-carbonitrile
2-(4-methyl-1H-pyrazol-1-yl)-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}acetamide
({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(6-methylpyridin-2-yl)methyl]amine
1-[2-(morpholin-4-yl)ethyl]-4-(1,2-oxazole-3-carbonyl)-1,4-diazepan-6-ol
2-[5-(2H-1,2,3-benzotriazol-2-ylmethyl)-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
2-(dimethylamino)-N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-4-methylpyrimidine-5-carboxamide
5-{[({4-[(2-methoxyethyl)carbamoyl]phenyl}carbamoyl)amino]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4-methyl-1H-imidazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(pyridazine-3-carbonyl)-N-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-{[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}benzonitrile
1-benzyl-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
8-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[(3-chloro-4,5-dimethoxyphenyl)methyl](methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-one
3-{2-[4-(3,4-difluorobenzoyl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-{1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}pyrrolidin-2-one
N-methyl-N-[2-(4-methylphenoxy)ethyl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
5-{[methyl(2-phenylethyl)amino]methyl}-N-(2-methylbutan-2-yl)-1,2-oxazole-3-carboxamide
3-(2-oxo-2-{4-[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]piperidin-1-yl}ethyl)-1,2,3-oxadiazol-3-ium-5-olate
1-[2-({[5-(2-chlorophenyl)furan-2-yl]methyl}(methyl)amino)ethyl]-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-1-[1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]piperidine-4-carboxamide
4-acetyl-5-benzyl-1-(4-methylphenyl)piperazin-2-one
1-(1H-imidazol-4-ylmethyl)-8-[8-(trifluoromethyl)quinolin-4-yl]-1,8-diazaspiro[4.5]decane
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-methoxyethan-1-one
5-cyclopropanecarbonyl-1'-(1,4-dithiepan-6-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(azocan-1-yl)-1-{4-[2-(2-hydroxyethoxy)ethyl]piperazin-1-yl}propan-1-one
1-(cyclohexylmethyl)-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
1-(2-chloro-4,6-dimethylphenyl)-3-cyclopropyl-3-(1,3-thiazol-2-ylmethyl)urea
1-acetyl-N-[(3-phenylphenyl)methyl]piperidine-3-carboxamide
methyl 3-cyclobutaneamido-5-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
4-methoxy-6-[3-(piperidin-1-yl)azetidin-1-yl]pyrimidine
N-cyclopentyl-2-({[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}amino)propanamide
1-{1,3-dioxo-2-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-isoindol-4-yl}-N-[1-(thiophen-2-yl)ethyl]piperidine-4-carboxamide
(1R,5R)-6-benzyl-3-(3,5-difluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonane
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(4-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
N-(1-ethyl-1H-indazol-3-yl)-2-[4-(1-methyl-1H-imidazol-2-yl)-1H-pyrazol-1-yl]acetamide
4-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-2-ethyl-1-(propan-2-yl)piperazine
2-{5-[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol