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4-{3-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyridin-2-yl}morpholine
4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}-N-(pyridin-4-ylmethyl)benzamide
1-(4-chloro-2,6-dimethylphenyl)-3-methyl-3-[(4-methyl-1H-imidazol-2-yl)methyl]urea
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-1-cyclohexyl-N-methylpiperidine-4-carboxamide
1-{8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]{2-[(4-methylphenyl)sulfanyl]propyl}amine
[(3R,4R)-4-(pyrrolidin-1-ylmethyl)-1-(quinoxalin-2-yl)pyrrolidin-3-yl]methanol
4-{4-[2-(4-chloro-2-methylphenoxy)propanoyl]piperazin-1-yl}-2-[2-(4-fluorophenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
5-(morpholine-4-carbonyl)-2-[2-(piperidin-1-yl)ethyl]-2,3-dihydro-1H-isoindol-1-one
7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-[(3S,4R)-3-cyclopropyl-4-[(pyrimidin-2-yl)amino]pyrrolidin-1-yl]-1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]ethan-1-one
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-1-(carbamoylmethyl)piperidine-4-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(oxan-4-yl)-5-(1,2-oxazol-3-yl)-1H-1,2,4-triazole
3-(2-phenylethyl)-8-(1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(4-methoxyphenyl)methyl]-8-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl](methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
1-tert-butyl-3-(oxan-4-yl)-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,4-triazole
1-[3-(furan-2-yl)propanoyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-fluoro-5-sulfamoylbenzamide
2-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
N3-cyclooctyl-N5-[(2,6-difluoro-3-methylphenyl)methyl]-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(2S,4R)-4-amino-N,N-diethyl-1-(2-methoxypyrimidine-5-carbonyl)pyrrolidine-2-carboxamide
3-chloro-N-[(2S)-1-hydroxypropan-2-yl]-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
1-[(2-fluorophenyl)methyl]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
5-[(5-ethylpyridin-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
1-(propan-2-yl)-4-(1H-pyrazole-4-carbonyl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
1-{2-[3-(2-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}-5-methylpyrrolidin-2-one
N-ethyl-3-methoxy-N-[(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)methyl]propanamide
N-(2-fluorophenyl)-3-[2-(pyridin-2-yl)acetamido]propanamide
2-ethyl-N-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-2H-1,2,3,4-tetrazol-5-amine
1-[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
[(4aS,8aR)-6-(5-fluoro-3,8-dimethylquinolin-2-yl)-decahydro-1,6-naphthyridin-4a-yl]methanol
(1R,9aR)-1-({[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]amino}methyl)-octahydro-1H-quinolizin-1-ol
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-(3-methoxyphenyl)-3-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}propanamide
(3S,4S)-4-cyclopropyl-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]pyrrolidine-3-carboxylic acid
(3S,4S)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-(9H-fluoren-9-yl)-5-methyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
1-{2-[1-(2,6-difluoro-4-methoxybenzoyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-oxoimidazolidin-1-yl)acetamide
2-methyl-4-phenyl-N-(1,3,4-thiadiazol-2-yl)piperazine-1-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(3-methoxypropyl)piperidin-1-yl]propan-1-one
4-(6-chloro-2-methylquinoline-4-carbonyl)-3-(propan-2-yl)piperazin-2-one
6-methyl-2-{[methyl({2-[(4-methylphenyl)sulfanyl]ethyl})amino]methyl}pyridin-3-ol
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-(2-methylpentyl)piperidine
7-fluoro-N,2-dimethyl-N-(1-methylpyrrolidin-3-yl)quinoline-4-carboxamide
1-methyl-3-(2-methylpropyl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
4-benzyl-1-(2-chlorobenzoyl)-3-ethyl-1,4-diazepan-5-one
(3R,4R)-1-[(3-ethoxy-4-hydroxyphenyl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol