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2-cyclopropyl-4-phenyl-9-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-amino-1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]hexan-1-one
5-ethyl-N-[4-(pyridin-2-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-(propane-1-sulfonyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-(3-methoxyphenyl)-4-[3-(pyrrolidin-1-yl)piperidin-1-yl]piperidine
5-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(2-methoxyphenyl)methyl]-N-methyl-1H-pyrazole-3-carboxamide
2-(1H-pyrazol-1-yl)-1-[4-(thian-4-yl)piperazin-1-yl]butan-1-one
N-[3-(3-chlorophenyl)phenyl]-1-(1,2,3-thiadiazole-4-carbonyl)piperidine-4-carboxamide
N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)quinoline-6-carboxamide
2-methyl-N-[2-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)ethyl]-1,3-thiazole-4-carboxamide
3-[(3R,4S)-1-[(5-methylthiophen-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-[2-(1H-indol-1-yl)ethyl]-3-(1H-1,2,3,4-tetrazol-5-yl)urea
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-6-(propan-2-yl)pyrimidin-4-amine
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(thiophene-2-carbonyl)pyrrolidin-3-yl]-1H-1,2,4-triazole-5-carboxamide
3-[N-(2-phenylethyl)-1-[4-(1H-pyrazol-3-yl)phenyl]formamido]propanamide
1-[(4-methoxyphenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
5-ethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
(1s,4s)-4-hydroxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]cyclohexane-1-carboxamide
N-(2-methoxyphenyl)-3-{[4-(methylamino)pyrimidin-2-yl]amino}propanamide
3-(3-fluorophenyl)-N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
3-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
1-(3-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}phenyl)ethan-1-one
(4aS,7aR)-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(azocan-1-yl)-3-[2-methoxy-4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-{[(1-methyl-1H-imidazol-2-yl)methyl]({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})amino}ethan-1-ol
ethyl 3-benzyl-1-(4-acetamidobenzenesulfonyl)piperidine-3-carboxylate
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-methylpropanamide
1-(1-benzylpiperidin-4-yl)-N-tert-butylpiperidine-3-carboxamide
(1H-1,3-benzodiazol-2-ylmethyl)[2-(2-ethoxyphenoxy)ethyl]methylamine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3,5-dicarboxamide
6-(2-chlorophenyl)-N-(2-fluoroethyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-[(2S)-1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
(1R,5R)-N,N-dimethyl-6-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-ethoxy-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyridine-3-carboxamide
3-{[(5-chloro-2,4-dimethoxyphenyl)methyl](methyl)amino}-N-methylbutanamide
N-(5-chloro-2-methoxyphenyl)-3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidine-1-carboxamide
4-(4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
2-methoxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-sulfamoylbenzamide
methyl 3-{[(4-fluorophenyl)formamido]methyl}-5-(furan-2-amido)benzoate
2-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(4-hydroxypiperidin-1-yl)acetamide
3-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-5-(2,6-difluorophenoxymethyl)-1,2-oxazole
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-5-{1-[(3E)-pent-3-enoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
(2S,4S)-4-amino-N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-methylpyrrolidine-2-carboxamide
{1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
2-[1-oxo-1-(3-oxo-4-phenylpiperazin-1-yl)butan-2-yl]-2,3-dihydro-1H-isoindol-1-one
N-(2-methoxyethyl)-4-methyl-N-{[2-(2-methylphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}benzamide
N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(4H-1,2,4-triazol-4-yl)benzamide