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2-(dimethylamino)-2-(3-methylphenyl)-1-{1-oxa-7-azaspiro[3.5]nonan-7-yl}ethan-1-one
N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-4-sulfamoylbenzamide
5-(pyrrolidin-2-yl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]thiophene-2-carboxamide
5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1H-pyrazole-4-carboxamide
(3R,9aR)-8-[(2-fluorophenyl)methyl]-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl (1R,3S,3aR,6aS)-3-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-{3-[methyl(phenyl)amino]propyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-propylbenzamide
2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
N-cyclopentyl-2-[6-oxo-4-(piperazin-1-yl)-1,6-dihydropyridazin-1-yl]butanamide
5-methyl-1-(3-{[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methoxy}phenyl)-1H-1,2,3,4-tetrazole
1-{[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazol-5-amine
[(3R,4R)-1-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
1-(cyclohexylmethyl)-6-oxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidine-3-carboxamide
5-{2-[2-({5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}amino)ethyl]morpholin-4-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-phenyl-3-({1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}formamido)propanamide
3-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-8-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]methylamine
2-[2-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyridine
methyl 6-[(3,4-dimethylphenyl)methyl]-2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(1-benzofuran-2-ylmethyl)-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-amine
7-(2-methoxyphenyl)-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepine-2-carboxamide
N-cyclopropyl-5-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-methylbenzamide
3-(2-ethoxyethoxy)-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)benzamide
3-(4-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}piperazin-1-yl)-1,2-benzothiazole
3-[1-ethyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]-3,4-dihydro-2H-1λ6,2-benzothiazine-1,1-dione
5-fluoro-N-[3-(pyridin-4-yl)propyl]quinazolin-4-amine
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
(1S,5R)-6-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
7-(3-hydroxy-2-methylbenzoyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(2,6-difluorophenyl)ethan-1-one
5-(3-methyl-1,2,4-oxadiazol-5-yl)-2-{3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyridine
3-(2H-1,3-benzodioxol-5-ylmethyl)-7-fluoro-3,4-dihydroquinazolin-4-one
4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide
4-{[1-(but-2-ynoyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-[methyl(phenyl)amino]ethan-1-one
7-[2-(oxan-2-ylmethoxy)acetyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
7-(5-chloropyridin-2-yl)-4-(pyrazin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
(3S)-4-(2,6-difluoro-4-methoxybenzoyl)-3-ethylmorpholine
1-(5-chloro-2-methoxyphenyl)-3-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-3-methylurea
(4R)-4-{3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1,3-thiazolidin-2-one
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
3-(2-methyl-1H-imidazol-1-yl)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]propanamide