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(3S,4S)-1-[benzyl(methyl)sulfamoyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]acetamide
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]propan-1-one
1-cyclohexyl-5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-3-(2-methoxyethyl)-1H-1,2,4-triazole
1-[(2-chloro-4-fluorophenyl)methyl]-N-[(3-methoxyphenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-(4-fluorophenyl)-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-hydroxyethan-1-one
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
2-(4-fluorophenyl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-cyclopropyl-1-[1-(pyridine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-(2-hydroxyethyl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
4-(3-cyanophenyl)-N-(4-methanesulfonylphenyl)piperidine-1-carboxamide
7-(5-chloro-2-methoxyphenyl)-4-[(2-fluorophenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-{2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-1H-1,2,3,4-tetrazole
7-(1,3-benzothiazol-2-yl)-4-[1-(methoxymethyl)cyclopropanecarbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2-methyl-1H-indol-3-yl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
3-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(1R)-1-phenylpropyl]urea
(2S,4S)-1-benzyl-N-ethyl-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
2-{[2-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-[2-(trifluoromethyl)phenyl]acetamide
N-({1-[(3-ethenylphenyl)methyl]piperidin-3-yl}methyl)-2-hydroxyacetamide
4-[4-(1H-imidazole-2-carbonyl)phenyl]-1-methyl-1H-pyrazole
N-{2-[2-(trifluoromethyl)phenyl]ethyl}pyrimidin-2-amine
(3R,4R)-3,4-dimethyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-ol
ethyl 3-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}butanoate
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-2-cyclopropyl-4-hydroxypyrimidine-5-carboxamide
3-{2-oxo-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
3-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-3-(furan-2-yl)-3-phenylpropan-1-one
1-phenyl-4-[1-(2-phenylethyl)piperidin-3-yl]piperazine
N-[3-(2-ethoxyphenyl)propyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
5-methoxy-1,2-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-indole-3-carboxamide
2-methyl-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}quinolin-4-amine
2-[4-(4-methanesulfonylpiperazin-1-yl)-5,6-dimethylthieno[2,3-d]pyrimidin-2-yl]ethan-1-amine
1-(4-benzylpiperazine-1-carbonyl)-6-[5-(methoxymethyl)furan-2-carbonyl]-6-azaspiro[2.5]octane
3-(1-benzyl-1H-imidazol-2-yl)-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
N-(2-methylpropyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
N-(1H-indol-2-ylmethyl)-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{2-[(2-chlorophenyl)methyl]morpholine-4-carbonyl}pyridin-2-ol
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(pyrrolidin-1-yl)piperidine
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
6-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carboxamide
3-(azepane-1-carbonyl)-N-(cyclopropylmethyl)-1-(prop-2-en-1-yl)-N-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{2-[7-(5-chloro-2-methoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-4-phenylpyrrolidin-2-one
methyl 4-{4-[2-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]piperazin-1-yl}benzoate