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methyl (2R,4S)-4-hydroxy-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine-2-carboxylate
ethyl 5-[(4-hydroxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
methyl 3-{[(1-methylazepan-2-yl)formamido]methyl}-5-[(2E)-3-phenylprop-2-enamido]benzoate
2-[2-(4-fluorophenoxy)ethyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-(1,3-benzothiazol-2-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(2R)-2-amino-N-(cyclohex-1-en-1-ylmethyl)-2-phenylacetamide
2-{[6-(1H-pyrazol-3-yl)quinazolin-4-yl]amino}ethan-1-ol
4-(1-ethyl-1H-1,3-benzodiazol-2-yl)-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(3S,4S)-4-cyclopropyl-1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidine-3-carboxylic acid
3-{4-[1-(2-methoxyethyl)piperidine-4-carbonyl]piperazin-1-yl}phenol
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-N-methylpiperidine-2-carboxamide
methyl (2S,4S)-1-[(2,4-difluorophenyl)methyl]-4-(2-fluorobenzamido)pyrrolidine-2-carboxylate
3-cyclopropyl-1-ethyl-5-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
1-(3,3-diphenylpiperidin-1-yl)-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
4-[3-(3-methoxybenzoyl)piperidin-1-yl]-6-(propan-2-yl)pyrimidine
N1,N1-dimethyl-N3-[(4-sulfamoylphenyl)methyl]piperidine-1,3-dicarboxamide
5-(1-methyl-1H-imidazol-2-yl)-1-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-4-phenyl-1H-imidazole
5-methyl-2-(methylamino)-N-[2-(1-methylpiperidin-3-yl)ethyl]benzamide
N-[(5-{[5-(2-fluorophenyl)furan-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
1-[4-(4-methylphenoxy)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
[(3S,5R)-5-[(dimethylamino)methyl]-1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-3-yl]methanol
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2,3-dimethyl-1H-indole-5-carboxamide
2-chloro-4-{[4-(5-ethyl-2-methylpyrimidin-4-yl)piperazin-1-yl]methyl}-6-methoxyphenol
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-benzyl-3-methyl-4-(3-methyl-1H-pyrazol-5-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-(2-methylphenyl)acetyl]pyrrolidin-3-yl]acetamide
4-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]benzene-1-sulfonamide
2,6-dihydroxy-N-[1-(pyridin-3-ylmethyl)piperidin-3-yl]benzamide
N-[(2S)-4-(methylsulfanyl)-1-oxo-1-(3-oxo-4-phenylpiperazin-1-yl)butan-2-yl]acetamide
N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
[(3R,5R)-1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
1-ethyl-5-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}-1H-indole
methyl 3-[(2E)-3-(3-fluorophenyl)prop-2-enamido]-6-[(4-formyl-1,4-diazepan-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(piperidin-1-yl)acetamide
2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoxaline
2-(1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
N-(furan-2-ylmethyl)-6,6-dimethyl-5-oxo-N-(2-phenylethyl)thiomorpholine-3-carboxamide
5-[1-(2-cyclohexylacetyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(6-ethyl-2-methylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
6-{2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}pyridine-2-carbonitrile
1-(4-aminopyrimidin-2-yl)-4-(oxan-4-yl)-1,4-diazepan-6-ol
N-methyl-N-(2-phenylethyl)-1-phenylmethanesulfonylpiperidin-3-amine
1-(pyridazine-3-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
5-[7-(3-methoxyphenyl)-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl]-N,N-dimethylfuran-2-carboxamide
1-methyl-4-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methoxypyrimidine
N-butyl-5-[2-(hydroxymethyl)phenyl]furan-2-carboxamide
[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]methanol