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7-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decane
7a-{2-[4-(1-phenylethyl)-1H-1,2,3-triazol-1-yl]ethyl}-hexahydro-1H-pyrrolizine
1-(5-chloropyridin-2-yl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylic acid
1-cyclohexyl-N5-cyclopropyl-N3-methyl-4-oxo-N3-(quinolin-5-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-amino-3-phenylpropanamide
1-[(1s,4s)-4-aminocyclohexyl]-N-(1,2,3,4-tetrahydronaphthalen-2-yl)-1H-1,2,3-triazole-4-carboxamide
7-methoxy-N,N-dimethyl-2-[1-(2-methylpyridin-4-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-(2-fluoroethyl)-3-{[1-(4-fluorophenyl)ethyl](methyl)sulfamoyl}benzamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-3-yl]methanol
3,4,7-trimethyl-2-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}-1H-indole
2-(3,4-dichlorophenyl)-4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]morpholine
methyl[1-(3-methylpyridin-2-yl)propan-2-yl]{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-[3-(2-hydroxypropan-2-yl)pyrrolidine-1-carbonyl]-5-methoxyphenol
(4aS,7aR)-1-(2-hydroxybenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1-methyl-1H-imidazol-2-yl)({1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl})methanol
2-(2-ethyl-1H-imidazol-1-yl)-1-[2-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
4-[(2S)-1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}pyrrolidine-2-carbonyl]morpholine
8-(3-ethoxypropanoyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
5-methyl-4-{2-oxo-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydro-1H-pyrazol-3-one
(4aS,8aR)-6-(4-aminopyrimidin-2-yl)-1-(carboxymethyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-[2-(3-fluorophenyl)ethyl]-2-[4-(4-{[1-(1,3-thiazol-5-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]acetamide
3-(3-{3-[cyclohexyl(methyl)amino]propyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)propanamide
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidin-3-amine
(4aR,7aS)-1-benzyl-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-phenylphenyl)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1H-imidazole
1-[(2,5-dimethylphenyl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(1S,5R)-6-(5-chlorothiophene-2-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[4-(naphthalen-2-yl)piperazin-1-yl]-4-oxobutane-1-sulfonamide
6-{[(cyclopropylmethyl)(propyl)amino]methyl}-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
(3R,4R)-1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-3,4-dimethylpyrrolidin-3-ol
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[(1S,2R)-2-(hydroxymethyl)cyclopentyl]benzamide
2-methoxy-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}isoquinoline
N,N-diethyl-15-methyl-13-oxo-9-(pyridin-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
6-cyclopentyl-2-methoxy-3-{[(5-propylpyrimidin-4-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
2-{[(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}phenol
2-(2-methyl-1,3-thiazol-4-yl)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}acetamide
(1R,5R)-3-(3-chloro-1H-indole-2-carbonyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-({2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxyphenyl}formamido)acetamide
N-[1-(2,5-dimethylphenyl)ethyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetamide
(4aS,8aR)-6-[(3-fluoro-4-methoxyphenyl)methyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
7-{[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]methyl}-2-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
2-amino-3-ethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-(2-fluoro-4-methylphenyl)-4-[2-(methylsulfanyl)ethyl]piperazine-1-carboxamide
1-{3-[3-(4-methylphenoxymethyl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
(2S,4R)-N-methyl-4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
(4aS,7aR)-1-(pyridine-3-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione