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5-[2-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-oxoethyl]-2,6-dimethyl-3,4-dihydropyrimidin-4-one
2-[1-(2-methylpropyl)-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-2-yl]ethan-1-ol
3-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
3,3-dimethyl-1-[(3S,5S)-1-methyl-5-(4-methylpiperazine-1-carbonyl)pyrrolidin-3-yl]urea
2-[4-({[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)amino}methyl)phenyl]-6-propyl-3,4-dihydropyrimidin-4-one
3-[(3R,4S)-4-(dimethylamino)-1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)piperidin-3-yl]propan-1-ol
N-methyl-N-[2-(4-methylphenoxy)ethyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carboxamide
(1H-indol-4-ylmethyl)(methyl)[2-(oxan-2-yl)ethyl]amine
2-(dimethylamino)-1-[3-(2-fluorophenoxy)azetidin-1-yl]-2-(2-fluorophenyl)ethan-1-one
1-(dimethylcarbamoyl)-4-[6-(methylcarbamoyl)pyridin-2-yl]-1,4-diazepane-6-carboxylic acid
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-{2-[2-(4-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
3-[1-(2-benzyl-1,3-thiazole-4-carbonyl)azetidin-3-yl]pyridine
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-2-(pyridin-2-yl)acetamide
2-ethyl-9-[(2,3,5,6-tetrafluoro-4-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(3-hydroxy-3-methylbutyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]benzamide
N,N-bis(furan-2-ylmethyl)-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
1-{4-[(3S,4S)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
2-{1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]pyrrolidin-3-yl}benzoic acid
2-methyl-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-3-(1H-1,2,4-triazol-1-yl)propanamide
N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-methoxy-N-{3-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]-3-oxopropyl}benzamide
(1S,5R)-3-[5-(propan-2-yl)pyrimidin-4-yl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methanesulfonylethyl)-3,4,7-trimethyl-1H-indole-2-carboxamide
3-(1,3-benzothiazol-2-yl)-1-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]propan-1-one
5-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}isoquinoline
(4aR,7aS)-1-(2,2-dimethylpropanoyl)-4-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-{1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-4-yl}phenyl)ethan-1-one
8-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylbenzamide
7-(cyclobutylmethyl)-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-methyl-N-{3-[methyl(phenyl)amino]propyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)pyridine-2-carboxamide
N-{1-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylcyclopropanecarboxamide
2-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(2,5-dimethoxyphenyl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenol
3-fluoro-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
3-[(4aR,7aS)-4-(3-methoxybenzoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-[(2-fluorophenyl)methyl]-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-(2-hydroxyethyl)acetamide
8-(2-aminoacetyl)-3-{2-[methyl(2-phenylethyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(4-methoxy-2,5-dimethylphenyl)methyl]methylamine
2-amino-4-(2-methoxypyrimidin-5-yl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
(3aS,6aS)-2-(2-methoxyacetyl)-5-{[3-(methylsulfanyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
(3aS,6aS)-5-[2-(2,3-dimethylphenoxy)ethyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5,7-dimethyl-N-[3-methyl-2-(pyrrolidin-1-yl)butyl]pyrido[2,3-d]pyrimidin-4-amine
1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-3-(thiophen-3-yl)propan-1-one
N-(3-{6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-3-oxopropyl)-4-methylbenzamide
N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-1H-pyrazole-5-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[3-(3-methylphenyl)phenyl]pyrrolidine-2-carboxamide