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3-[1-(2,5-dimethoxyphenyl)-1H-imidazol-2-yl]phenol
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]acetamide
(1R,5R)-N-(2,4-dichlorophenyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
methyl 1-[(3R,5S)-5-[(diphenylmethyl)carbamoyl]-1-[(3-methoxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5,7-dimethyl-3-[3-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-[1,2,4]triazolo[4,3-a]pyrimidine
7-(2-methoxypyridine-4-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-2-methylpyrido[2,3-d]pyrimidin-4-amine
N,2-dimethyl-N-{2-phenyl-1-[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]ethyl}furan-3-carboxamide
4-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-N-methylpyridin-2-amine
methyl 6-(2,3-dihydro-1-benzofuran-2-carbonyl)-2-[(3-methylbutyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(3-fluoropyridin-2-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-3-[(3-methylthiophen-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-(propan-2-yloxy)pyrimidin-2-amine
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-2-(methylamino)pyridine-4-carboxamide
1-cyclopentyl-N-phenylpiperidin-3-amine
N-{2-[2-methyl-5-(morpholine-4-sulfonyl)-1H-1,3-benzodiazol-1-yl]ethyl}-2-(methylsulfanyl)acetamide
1,3-dimethyl-6-{1-oxa-8-azaspiro[4.6]undecane-8-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-benzyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1,3-thiazole-4-carboxamide
3-(1-ethyl-1H-imidazol-2-yl)-1-(4-methoxybenzoyl)piperidine
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
2-(4-{4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}piperazin-1-yl)ethan-1-ol
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}benzamide
1-(4-carbamoylpyridin-2-yl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
3-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}phenol
[5-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)furan-2-yl]methanol
3-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroisoquinolin-1-one
3-[4-(3-hydroxyphenyl)piperidin-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
3-[2-chloro-5-(morpholine-4-carbonyl)phenyl]-1-(oxan-4-yl)urea
2-{2-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-6-methyl-2,3-dihydropyridazin-3-one
{1-[5-(2-chlorophenyl)-2-methylfuran-3-carbonyl]piperidin-2-yl}methanol
1-(1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)ethan-1-one
(2S,4S)-N-ethyl-4-[2-(pyridin-3-yl)acetamido]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N-(furan-2-ylmethyl)-N-methyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
3-fluoro-5-[6-(hydroxymethyl)-1,4-oxazepane-4-carbonyl]benzonitrile
2-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}methyl)-3,4-dihydroquinazolin-4-one
ethyl 3-benzyl-1-{[1-(carbamoylmethyl)-1H-indol-3-yl]methyl}piperidine-3-carboxylate
N-[3-(cyclohexyloxy)propyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[3-(trifluoromethyl)phenyl]piperazine
2-cyclobutyl-N-[(3R,4S)-4-cyclopropyl-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]acetamide
[(3R,5R)-5-[(dimethylamino)methyl]-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-3-yl]methanol
N-[1-(furan-2-carbonyl)piperidin-3-yl]-2-methyl-5-propylpyrimidin-4-amine
3-[2-(3-fluorophenyl)ethyl]-1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}piperidine
3-(azepane-1-carbonyl)-1-ethyl-N-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetamide
N-[2-(diethylamino)ethyl]-N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-(2-chlorophenyl)-3-[1-(furan-3-ylmethyl)piperidin-4-yl]propanamide
4-amino-11-hydroxy-6-[2-(2-hydroxyethoxy)phenyl]-8-oxa-3-azatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaene-5-carbonitrile
1-(2-methylquinolin-5-yl)-3-[4-(oxolan-2-yl)butyl]urea