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3-[1-(2,6-dimethylpyridin-4-yl)-N-methylformamido]-N-methylbutanamide
3-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)azetidin-3-yl]pyridine
4-(3-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidine-1-carbonyl}phenyl)-2-methylbutan-2-ol
1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-4-[(3,5-difluorophenyl)methyl]piperazine
2,3,6-trimethyl-4-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carbonyl]quinoline
2,2-dimethyl-N-[4-methyl-3-(4-methylbenzamido)phenyl]oxane-4-carboxamide
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
7-[(3,3-difluoropyrrolidin-1-yl)methyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1-ethyl-3,5-dimethyl-4-[3-methyl-1-(4-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
(1S,5R)-3-(1-benzylpiperidin-4-yl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
N,5-dimethyl-N-(1-methylpiperidin-4-yl)-4-[(3-phenylpropyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-1-methyl-5-phenyl-1H-pyrrole
(3S,4R)-1-(4-chloro-2-hydroxybenzoyl)-4-methylpiperidine-3,4-diol
2-[1-(2-phenylethyl)-4-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl]ethan-1-ol
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-3-methylbut-2-en-1-one
N-(3-hydroxy-3-phenylpropyl)-N-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
(1R,5R)-6-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-methyl-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[1-(4-methylpyridin-2-yl)propyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
1-(1H-pyrrole-2-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
4-(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
(3R,4R)-3-cyclobutyl-4-methyl-1-[5-(morpholine-4-carbonyl)pyridin-2-yl]pyrrolidin-3-ol
2-(pyridin-3-yl)-7-[2-(1H-1,2,4-triazol-3-ylsulfanyl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[7-chloro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]cyclobutanecarboxamide
6-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}pyridine-3-carboxamide
4-(hydroxymethyl)-N,N-dimethyl-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-1-sulfonamide
4-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-cyclohexylpiperazin-2-one
3-(4-methanesulfonylphenyl)-1H-indazole
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-(4-fluoro-3-methylphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-2,5-dimethylfuran-3-carboxamide
1-[(2,5-dimethylphenyl)methyl]-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-[2-(3-acetyl-1H-indol-1-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-methyl-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
2-{4-[(2-methylpyridin-3-yl)methyl]piperazin-1-yl}pyrazine
dimethyl({[4-(4-methylphthalazin-1-yl)phenyl]methyl})amine
4-[(4-fluorophenyl)methyl]-1-(6-methylpyridine-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(3aR,6aR)-2-cyclopropanecarbonyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
[1-({1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
benzyl(cyclopropylmethyl){[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
N-(1-methanesulfonylpiperidin-4-yl)-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-(3-methylbutyl)-8-(2,4,6-trimethylbenzoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-methyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)azepane-2-carboxamide
1-(2-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}ethyl)-1H-imidazole
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-(1H-indol-3-yl)butanamide
1-(cyclopent-1-ene-1-carbonyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
2-(3-fluoro-4-methoxyphenyl)-2-{methyl[(3-methylpyridin-4-yl)methyl]amino}acetic acid
N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
(3R,4R)-N-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carboxamide