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2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-(pyridin-4-ylmethyl)acetamide
4-(furan-2-carbonyl)-7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-cyclohexyl-2-[methyl(piperidin-4-yl)amino]-N-(pyridin-4-ylmethyl)acetamide
(3S,4R)-1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-1,3-thiazole-5-carboxamide
4-(3-chloro-5-fluoro-4-methoxyphenyl)-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole
4-[(4-hydroxyphenyl)methyl]-6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2,3-dihydro-1,4-benzodioxine-2-carboxamide
1-(3-chlorophenyl)-4-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]piperazin-2-one
(4aR,7aS)-1-cyclobutanecarbonyl-4-{[4-(propan-2-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2R,4R,6S)-2-(3,5-difluorophenyl)-6-[3-(propan-2-yl)-1,2-oxazol-5-yl]oxan-4-yl]acetamide
(2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
1,5-dimethyl-4-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-(5-fluoro-2-methylphenyl)-3-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)benzamide
2-methyl-5-(4-{[(2-methyl-5-propylpyrimidin-4-yl)amino]methyl}piperidin-1-yl)-2,3-dihydropyridazin-3-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(thian-4-yl)piperazin-2-yl}ethan-1-ol
1-(2-chlorophenyl)-5-methyl-4-[3-(piperidin-1-yl)propanoyl]piperazin-2-one
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-(3-methoxypropyl)-8-(quinoxalin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-benzyl-6-(3-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
8-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
3-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethyl-1-(4-methylphenyl)urea
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
3-(2,4-difluorophenyl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-butyl-4-(2,8-dimethylquinoline-4-carbonyl)-1-methylpiperazin-2-one
5-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-methyl-3-{[4-(3-propoxypiperidine-1-carbonyl)piperidin-4-yl]oxy}pyridine
3-[4-(dimethylamino)butyl]-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
2-(3-hydroxyphenyl)-1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
2-{4-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]piperidin-1-yl}pyrazine
N-[2-(2-chlorophenyl)-1-[1-(quinolin-7-ylmethyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
N-[3-({[1-(1H-imidazol-1-yl)butan-2-yl]carbamoyl}amino)phenyl]-2-methoxyacetamide
1-benzyl-5-[(2,3-dihydro-1H-inden-2-yl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(3-oxo-4-phenylpiperazine-1-carbonyl)cyclopropane-1-carboxamide
5-{2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
1-[(4-fluorophenyl)methyl]-4-({[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}amino)pyrrolidin-2-one
2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}quinoline
4-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-2-methylphenol
N-(1,4-dioxan-2-ylmethyl)-N-methyl-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
methyl 5-cyano-6-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-methylpyridine-3-carboxylate
5-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole
N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)oxolane-3-carboxamide
(3R,4R)-3,4-dimethyl-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)pyrrolidin-3-ol
4-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide