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5-fluoro-N2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N4,N4-dimethylpyrimidine-2,4-diamine
1-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
1-({3-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]phenyl}methyl)-1H-pyrazole
4-(3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propanoyl)-6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-1,4-diazepan-2-one
1-benzyl-5-(4-cyclohexylpiperazine-1-carbonyl)-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
8-methoxy-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(2-fluoro-6-methoxyphenyl)-5-methylpyridin-2-amine
2-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]-4-(trifluoromethyl)pyrimidine
N-butyl-3-[(4-hydroxypiperidin-1-yl)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
ethyl 3-({3-[(1H-indol-2-ylformamido)methyl]piperidine-1-carbonyl}amino)propanoate
[(3S,5R)-1-{[2-(difluoromethoxy)phenyl]methyl}-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
(3aR,5S,6S,7aS)-5,6-dihydroxy-N-{3-[(2-methylpropyl)carbamoyl]phenyl}-octahydro-1H-isoindole-2-carboxamide
1-[3-(pyrrolidin-1-yl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
N,N-dimethyl-3-(4-phenyl-1,4-diazepane-1-carbonyl)piperidine-1-carboxamide
2-{[(2,5-dimethylfuran-3-yl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
4-ethyl-3-(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[benzyl(methyl)amino]-2-[(2,3-dimethoxyphenyl)methyl]-2,3-dihydropyridazin-3-one
4-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
1-ethyl-5-methyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H-pyrazole-4-carboxamide
2-amino-6-(2-methylpropyl)-N-[2-phenyl-2-(piperidin-1-yl)ethyl]pyrimidine-4-carboxamide
1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-4-hydroxypiperidine-4-carboxylic acid
N-(furan-2-ylmethyl)-3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propanamide
4-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]piperazine-1-sulfonamide
2-methoxy-N-[4-methyl-3-({[3-(4-methyl-1,3-thiazol-2-yl)propyl]carbamoyl}amino)phenyl]acetamide
N-(3-chloro-4-propanamidophenyl)-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
6-(aminomethyl)-2-(3-{[methyl(3-phenoxypropyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-({1-[3-(pyridin-3-yl)propanoyl]pyrrolidin-3-yl}methyl)benzamide
N-[(4-fluorophenyl)methyl]-N-methyl-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-{2-[4-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,3-triazol-1-yl]ethyl}-N-methylmethanesulfonamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)[(4-methyloxan-4-yl)methyl]amine
N,N-dimethyl-5-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}pyridin-2-amine
9-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[2-(furan-2-yl)ethyl]acetamide
4-[(1-propyl-1H-imidazol-2-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(carbamoylmethyl)-N-{[1-(4-fluorophenyl)cyclopentyl]methyl}piperidine-4-carboxamide
4-{[6-(dimethylamino)pyridin-3-yl]methyl}-3-(4-fluorophenyl)piperazin-2-one
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-(4H-1,2,4-triazol-4-yl)piperidine
2-{2-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one
N-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[2-(piperidin-1-yl)ethyl]quinoline-4-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[2-(methylcarbamoyl)pyrrolidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
ethyl 5-{[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
4-(2-{1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}ethyl)morpholine
4-(4-{[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]methyl}phenyl)but-3-yn-1-ol
2-benzyl-N-[(5-methylfuran-2-yl)methyl]-1,3-thiazole-4-carboxamide
2-[2-(4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-1-yl)ethoxy]ethan-1-ol
N-methyl-N-{4-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}methanesulfonamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide